Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT03110 , Mucosa-associated lymphoid tissue lymphoma translocation protein 1
Gene Name MALT1
Organism Homo sapiens, Human
Protein Classification Enzyme
Uniprot ID Q9UDY8
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT03110
 
Compound ID Compound Name Compound Formula
CP0074453
1-(3-chloropyridin-2-yl)-N-[5-chloro-6-(triazol-2-yl)pyridin-3-yl]piperidine-4-carboxamide
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C18H17Cl2N7O
 1
1
IC50 = 90 nM
   TI
   LI
   LO
   TS
CP0536081
1-(3-aminopyridin-2-yl)-N-[5-chloro-6-(triazol-2-yl)pyridin-3-yl]piperidine-4-carboxamide
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C18H19ClN8O
 1
1
IC50 = 90 nM
   TI
   LI
   LO
   TS
CP0359950
1-(3-aminopyridin-2-yl)-N-[3-chloro-4-(triazol-2-yl)phenyl]piperidine-4-carboxamide
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C19H20ClN7O
 1
1
IC50 = 110 nM
   TI
   LI
   LO
   TS
CP0389888
N-[3-chloro-4-[3-(methylcarbamoyl)-1,2,4-triazol-1-yl]phenyl]-1-(3-chloropyridin-2-yl)piperidine-4-carboxamide
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C21H21Cl2N7O2
 1
1
IC50 = 140 nM
   TI
   LI
   LO
   TS
CP0475290
N-(5-chloro-6-methoxypyridin-3-yl)-1-(3-chloropyridin-2-yl)piperidine-4-carboxamide
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C17H18Cl2N4O2
 1
1
IC50 = 190 nM
   TI
   LI
   LO
   TS
CP0261160
N-(3-chloro-4-fluorophenyl)-1-(3-chloropyrazin-2-yl)piperidine-4-carboxamide
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C16H15Cl2FN4O
 1
1
IC50 = 290 nM
   TI
   LI
   LO
   TS
CP0359945
1-(3-aminopyridin-2-yl)-N-(3-chloro-4-fluorophenyl)piperidine-4-carboxamide
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C17H18ClFN4O
 1
1
IC50 = 420 nM
   TI
   LI
   LO
   TS
CP0327620
N-[3-chloro-4-(3,5-dimethyl-1,2,4-triazol-1-yl)phenyl]-1-(3-nitropyridin-2-yl)piperidine-4-carboxamide
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C21H22ClN7O3
 1
1
IC50 = 640 nM
   TI
   LI
   LO
   TS
CP0261159
N-(3-chloro-4-fluorophenyl)-1-(3-chloropyridin-2-yl)piperidine-4-carboxamide
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C17H16Cl2FN3O
 1
1
IC50 = 1350 nM
   TI
   LI
   LO
   TS
CP0236381
N-(3-chlorophenyl)-1-(3-chloropyridin-2-yl)piperidine-4-carboxamide
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C17H17Cl2N3O
 1
1
IC50 = 1590 nM
   TI
   LI
   LO
   TS
CP0359944
N-(3-chloro-4-fluorophenyl)-1-(3-cyanopyridin-2-yl)piperidine-4-carboxamide
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C18H16ClFN4O
 1
1
IC50 = 2700 nM
   TI
   LI
   LO
   TS
CP0485574
1-(3-chloropyridin-2-yl)-N-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]piperidine-4-carboxamide
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C22H21ClF3N5O
 1
1
IC50 = 3000 nM
   TI
   LI
   LO
   TS
CP0086265
N-(3-chloro-4-fluorophenyl)-1-pyrimidin-2-ylpiperidine-4-carboxamide
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C16H16ClFN4O
 1
1
IC50 = 3100 nM
   TI
   LI
   LO
   TS
CP0327621
N-(3-chloro-4-fluorophenyl)-1-phenylpiperidine-4-carboxamide
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C18H18ClFN2O
 1
1
IC50 = 3200 nM
   TI
   LI
   LO
   TS
CP0359942
N-(3-chloro-4-methylphenyl)-1-(3-chloropyridin-2-yl)piperidine-4-carboxamide
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C18H19Cl2N3O
 1
1
IC50 = 3700 nM
   TI
   LI
   LO
   TS