| Compound ID |
Compound Name |
Compound Formula |
|
CP0398970
|
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Tyr
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|
C77H129N23O19
|
1
|
| 1 |
EC50 = 0.06 nM
|
|
|
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CP0398972
|
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Lys-Tyr
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|
C76H127N23O19
|
2
|
| 1 |
EC50 = 0.15 nM
|
|
|
| 2 |
EC50 = 26 nM
|
|
|
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CP0423355
|
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Fly-Tyr
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|
C96H137N23O23
|
1
|
| 1 |
EC50 = 0.92 nM
|
|
|
|
CP0423356
|
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Lys-Tyr-Fly
Show/Hide
|
C102H149N25O24
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0431898
|
Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Tyr
Show/Hide
|
C75H125N23O19
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0431771
|
Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Trp-Tyr
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|
C86H135N25O20
|
1
|
| 1 |
EC50 = 26 nM
|
|
|
|
CP0436332
|
Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Lys-Trp
Show/Hide
|
C76H124N24O18S
|
1
|
| 1 |
EC50 = 32 nM
|
|
|
|
CP0423354
|
Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Lys-Trp-Fly
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|
C102H146N26O23S
|
1
|
| 1 |
EC50 = 53 nM
|
|
|
|
CP0400098
|
5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-3,8-dimethyl-1,3,4-benzotriazepin-2-one
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|
C27H32N6O
|
2
|
| 1 |
Kd = 16.98 nM
|
|
|
| 2 |
Ki = 13.18 nM
|
|
|
|
CP0529718
|
5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-8-methyl-3-(6,7,8,9-tetrahydro-5H-benzo[7]annulen-7-yl)-1,3,4-benzotriazepin-2-one
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|
C37H42N6O
|
1
|
| 1 |
Ki = 0.912 nM
|
|
|
|
CP0529717
|
7-(benzylamino)-5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-3,8-dimethyl-1,3,4-benzotriazepin-2-one
Show/Hide
|
C34H39N7O
|
1
|
| 1 |
Ki = 1.445 nM
|
|
|
|
CP0465566
|
5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-3,8-dimethyl-7-phenylmethoxy-1,3,4-benzotriazepin-2-one
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|
C34H38N6O2
|
1
|
| 1 |
Ki = 1.82 nM
|
|
|
|
CP0495742
|
5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-8-methyl-3-propan-2-yl-1,3,4-benzotriazepin-2-one
Show/Hide
|
C29H36N6O
|
1
|
| 1 |
Ki = 3.548 nM
|
|
|
|
CP0465568
|
3-benzyl-5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-8-methyl-1,3,4-benzotriazepin-2-one
Show/Hide
|
C33H36N6O
|
1
|
| 1 |
Ki = 3.802 nM
|
|
|
|
CP0529716
|
5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-8-methyl-3-(oxan-4-yl)-1,3,4-benzotriazepin-2-one
Show/Hide
|
C31H38N6O2
|
1
|
| 1 |
Ki = 6.607 nM
|
|
|
|
CP0465567
|
5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-8-methyl-3-propyl-1,3,4-benzotriazepin-2-one
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|
C29H36N6O
|
1
|
| 1 |
Ki = 6.761 nM
|
|
|
|
CP0526946
|
1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-8-methyl-5-(oxan-4-yl)-3-(6,7,8,9-tetrahydro-5H-benzo[7]annulen-7-yl)-1,3,4-benzotriazepin-2-one
Show/Hide
|
C36H40N6O2
|
1
|
| 1 |
Ki = 6.761 nM
|
|
|
|
CP0465565
|
5-cyclohexyl-3-(3,4-dihydro-2H-1,5-benzodioxepin-3-yl)-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-8-methyl-1,3,4-benzotriazepin-2-one
Show/Hide
|
C35H38N6O3
|
1
|
| 1 |
Ki = 8.71 nM
|
|
|
|
CP0439763
|
5-cyclohexyl-1-[4-[3-(1H-imidazol-2-yl)propylamino]phenyl]-3,8-dimethyl-1,3,4-benzotriazepin-2-one
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|
C28H34N6O
|
1
|
| 1 |
Ki = 20.42 nM
|
|
|
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CP0501046
|
5-cyclohexyl-1-[4-(1H-imidazol-2-ylmethylamino)phenyl]-3,8-dimethyl-1,3,4-benzotriazepin-2-one
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|
C26H30N6O
|
1
|
| 1 |
Ki = 50.12 nM
|
|
|
|
CP0457965
|
3-benzyl-5-cyclohexyl-1-[4-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl]-8-methyl-1,3,4-benzotriazepin-2-one
Show/Hide
|
C31H34N6O
|
1
|
| 1 |
Ki = 70.79 nM
|
|
|
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CP0526945
|
5-cyclohexyl-1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-3-(2-methoxyethyl)-8-methyl-1,3,4-benzotriazepin-2-one
Show/Hide
|
C29H36N6O2
|
1
|
| 1 |
Ki = 83.18 nM
|
|
|
|
CP0536616
|
2-amino-N-[4-(3-benzyl-5-cyclohexyl-8-methyl-2-oxo-1,3,4-benzotriazepin-1-yl)phenyl]-3-methylbutanamide
Show/Hide
|
C33H39N5O2
|
1
|
| 1 |
Ki = 112.2 nM
|
|
|
|
CP0495743
|
2-[4-(3-benzyl-5-cyclohexyl-8-methyl-2-oxo-1,3,4-benzotriazepin-1-yl)phenyl]guanidine
Show/Hide
|
C29H32N6O
|
1
|
| 1 |
Ki = 154.88 nM
|
|
|
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CP0465569
|
3-benzyl-5-cyclohexyl-1-[4-(4,5-dihydro-1H-imidazol-2-ylamino)phenyl]-1,3,4-benzotriazepin-2-one
Show/Hide
|
C30H32N6O
|
1
|
| 1 |
Ki = 288.4 nM
|
|
|
|
CP0535169
|
2-amino-N-[4-(3-benzyl-5-cyclohexyl-2-oxo-1,3,4-benzotriazepin-1-yl)phenyl]-3-methylbutanamide
Show/Hide
|
C32H37N5O2
|
1
|
| 1 |
Ki = 380.19 nM
|
|
|
|
CP0505621
|
2-[4-[3-benzyl-5-(cyclohexylmethyl)-2-oxo-1,3,4-benzotriazepin-1-yl]phenyl]guanidine
Show/Hide
|
C29H32N6O
|
1
|
| 1 |
Ki = 562.34 nM
|
|
|
|
CP0448566
|
1-[4-[2-(1H-imidazol-2-yl)ethylamino]phenyl]-3,8-dimethyl-5-(oxan-4-yl)-1,3,4-benzotriazepin-2-one
Show/Hide
|
C26H30N6O2
|
1
|
| 1 |
Ki = 616.6 nM
|
|
|
|
CP0457966
|
2-amino-N-[4-(3-benzyl-5-cyclohexyl-2-oxo-1,3,4-benzotriazepin-1-yl)phenyl]acetamide
Show/Hide
|
C29H31N5O2
|
1
|
| 1 |
Ki = 676.08 nM
|
|
|
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CP0439751
|
2-[4-(3-benzyl-5-cyclohexyl-2-oxo-1,3,4-benzotriazepin-1-yl)phenyl]guanidine
Show/Hide
|
C28H30N6O
|
1
|
| 1 |
Ki = 707.95 nM
|
|
|
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CP0526947
|
2-[4-[[4-(3-benzyl-5-cyclohexyl-2-oxo-1,3,4-benzotriazepin-1-yl)phenyl]methyl]phenyl]guanidine
Show/Hide
|
C35H36N6O
|
1
|
| 1 |
Ki = 933.25 nM
|
|
|
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CP0526948
|
2-[3-(3-benzyl-5-cyclohexyl-2-oxo-1,3,4-benzotriazepin-1-yl)phenyl]guanidine
Show/Hide
|
C28H30N6O
|
1
|
| 1 |
Ki = 2818.38 nM
|
|
|
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CP0467249
|
2-[4-(3-benzyl-2-oxo-5-phenyl-1,3,4-benzotriazepin-1-yl)phenyl]guanidine
Show/Hide
|
C28H24N6O
|
1
|
| 1 |
Ki = 3388.44 nM
|
|
|
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CP0465570
|
4-(3-benzyl-5-cyclohexyl-2-oxo-1,3,4-benzotriazepin-1-yl)benzoic acid;(2R,3R,4R,5S)-6-(methylamino)hexane-1,2,3,4,5-pentol
Show/Hide
|
C28H27N3O3
|
1
|
| 1 |
Ki < 100000 nM
|
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