Brief Information of the Compound and Protein
Compound Name
2-[4-(3-benzyl-5-cyclohexyl-8-methyl-2-oxo-1,3,4-benzotriazepin-1-yl)phenyl]guanidine
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PubChem ID
CID: 23626400
SID: 46487097
Canonical SMILES
Cc1ccc2c(c1)N(c1ccc(NC(N)=N)cc1)C(=O)N(Cc1ccccc1)N=C2C1CCCCC1
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Compound Formula C29H32N6O
Compound Structure
Protein Name
Parathyroid hormone/parathyroid hormone-related peptide receptor
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Parathyroid hormone receptor
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Parathyroid hormone receptor
Uniprot ID
Q03431
Gene Name
PTH1R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 154.88 nM
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