Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT02449 , P2Y purinoceptor 12
Gene Name P2RY12
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q9H244
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT02449
 
Compound ID Compound Name Compound Formula
CP0429288
1-[2-[1'-(2,2-dimethylpropyl)spiro[2H-indole-3,4'-piperidine]-1-yl]phenyl]-3-[4-(trifluoromethoxy)phenyl]urea
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C31H35F3N4O2
 1
1
IC50 > 20000 nM
   TI
   LI
   LO
   TS
CP0066917
1-[2-(2-propan-2-ylphenoxy)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea
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C22H20F3N3O3
 1
1
Ki > 70000 nM
   TI
   LI
   LO
   TS
CP0205635
1-[2-(2-tert-butylphenyl)sulfanylpyridin-3-yl]-3-(4-methylphenyl)urea
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C23H25N3OS
 1
1
Ki > 70000 nM
   TI
   LI
   LO
   TS
CP0233597
1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-(4-tert-butylphenyl)urea
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C26H31N3O2
 1
1
Ki > 70000 nM
   TI
   LI
   LO
   TS
CP0233599
1-(4-tert-butylphenyl)-3-[2-(2-propan-2-ylphenoxy)pyridin-3-yl]urea
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C25H29N3O2
 1
1
Ki > 70000 nM
   TI
   LI
   LO
   TS
CP0241700
1-[2-(2-tert-butylphenoxy)pyridin-3-yl]-3-[4-(trifluoromethoxy)phenyl]urea
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C23H22F3N3O3
 1
1
Ki > 70000 nM
   TI
   LI
   LO
   TS
CP0481503
1-(2,4-difluorophenyl)-3-[2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl]urea
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C19H12F5N3O2
 1
1
Ki > 70000 nM
   TI
   LI
   LO
   TS