| Compound ID |
Compound Name |
Compound Formula |
|
CP0533094
|
N-(2-hydroxyethyl)-1-[6-[(3-methylphenyl)methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
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|
C23H24N4O2
|
1
|
| 1 |
EC50 = 90 nM
|
|
|
|
CP0465603
|
1-[6-[(3,5-dimethylphenyl)methyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
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|
C24H26N4O2
|
1
|
| 1 |
EC50 = 97 nM
|
|
|
|
CP0483735
|
N-(2-hydroxyethyl)-1-[6-[[3-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
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|
C23H21F3N4O2
|
1
|
| 1 |
EC50 = 101 nM
|
|
|
|
CP0469157
|
1-[6-[(3-fluorophenyl)methyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
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|
C22H21FN4O2
|
1
|
| 1 |
EC50 = 106 nM
|
|
|
|
CP0477825
|
N-(2-hydroxyethyl)-1-[6-[[4-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
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|
C23H21F3N4O2
|
1
|
| 1 |
EC50 = 109 nM
|
|
|
|
CP0562771
|
1-[6-[(3,5-difluorophenyl)methyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
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|
C22H20F2N4O2
|
1
|
| 1 |
EC50 = 115 nM
|
|
|
|
CP0469154
|
N-(2-hydroxyethyl)-1-[4-[[3-(trifluoromethyl)phenyl]methyl]pyridin-2-yl]-2,3-dihydroindole-4-carboxamide
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|
C24H22F3N3O2
|
1
|
| 1 |
EC50 = 119 nM
|
|
|
|
CP0575033
|
N-(2-hydroxyethyl)-1-[6-[[3-(trifluoromethoxy)phenyl]methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H21F3N4O3
|
1
|
| 1 |
EC50 = 131 nM
|
|
|
|
CP0135239
|
1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
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|
C23H20F4N4O2
|
1
|
| 1 |
EC50 = 135 nM
|
|
|
|
CP0552729
|
1-[5-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyridazin-3-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
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|
C23H20F4N4O2
|
1
|
| 1 |
EC50 = 158 nM
|
|
|
|
CP0533958
|
1-[4-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-2-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H20F4N4O2
|
1
|
| 1 |
EC50 = 186 nM
|
|
|
|
CP0552730
|
1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-N-(3-hydroxypropyl)-2,3-dihydroindole-4-carboxamide
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|
C24H22F4N4O2
|
1
|
| 1 |
EC50 = 275 nM
|
|
|
|
CP0557089
|
1-(6-benzylpyrimidin-4-yl)-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
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|
C22H22N4O2
|
1
|
| 1 |
EC50 = 292 nM
|
|
|
|
CP0469156
|
1-[4-[fluoro-[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-2-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
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|
C23H19F5N4O2
|
1
|
| 1 |
EC50 = 329 nM
|
|
|
|
CP0552731
|
1-[6-[fluoro-[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H19F5N4O2
|
1
|
| 1 |
EC50 = 330 nM
|
|
|
|
CP0573133
|
1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]-hydroxymethyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
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|
C23H20F4N4O3
|
1
|
| 1 |
EC50 = 338 nM
|
|
|
|
CP0548688
|
N-(1,3-dihydroxypropan-2-yl)-1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C24H22F4N4O3
|
1
|
| 1 |
EC50 = 346 nM
|
|
|
|
CP0531329
|
N-(2-hydroxyethyl)-1-[6-[(3-methoxyphenyl)methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H24N4O3
|
1
|
| 1 |
EC50 = 351 nM
|
|
|
|
CP0477824
|
N-(2-hydroxyethyl)-1-[6-[3-(trifluoromethyl)phenyl]sulfanylpyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
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|
C22H19F3N4O2S
|
1
|
| 1 |
EC50 = 371 nM
|
|
|
|
CP0548689
|
1-[2-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H20F4N4O2
|
1
|
| 1 |
EC50 = 373 nM
|
|
|
|
CP0469155
|
1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-N-(4-hydroxybutyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C25H24F4N4O2
|
1
|
| 1 |
EC50 = 399 nM
|
|
|
|
CP0483739
|
1-[4-[[3-fluoro-5-(trifluoromethyl)phenyl]-hydroxymethyl]pyrimidin-2-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H20F4N4O3
|
1
|
| 1 |
EC50 = 399 nM
|
|
|
|
CP0451612
|
N-(2-fluoroethyl)-1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H19F5N4O
|
1
|
| 1 |
EC50 = 431 nM
|
|
|
|
CP0557090
|
1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-N-(2-methoxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C24H22F4N4O2
|
1
|
| 1 |
EC50 = 489 nM
|
|
|
|
CP0550448
|
1-[6-[fluoro-[3-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H20F4N4O2
|
1
|
| 1 |
EC50 = 557 nM
|
|
|
|
CP0531330
|
N-(2-hydroxyethyl)-1-[6-[hydroxy-[3-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H21F3N4O3
|
1
|
| 1 |
EC50 = 560 nM
|
|
|
|
CP0495716
|
1-[4-chloro-5-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyridazin-3-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H19ClF4N4O2
|
1
|
| 1 |
EC50 = 565 nM
|
|
|
|
CP0573132
|
1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-N,N-bis(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C25H24F4N4O3
|
1
|
| 1 |
EC50 = 673 nM
|
|
|
|
CP0465605
|
N-(2-hydroxyethyl)-1-[6-[[2-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H21F3N4O2
|
1
|
| 1 |
EC50 = 711 nM
|
|
|
|
CP0483736
|
1-[5-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]-4-methylpyridazin-3-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C24H22F4N4O2
|
1
|
| 1 |
EC50 = 754 nM
|
|
|
|
CP0550447
|
[1-[6-[[3-fluoro-5-(trifluoromethyl)phenyl]methyl]pyrimidin-4-yl]-2,3-dihydroindol-4-yl]-(3-hydroxyazetidin-1-yl)methanone
Show/Hide
|
C24H20F4N4O2
|
1
|
| 1 |
EC50 = 760 nM
|
|
|
|
CP0495720
|
1-[6-[(3,5-dimethoxyphenyl)methyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C24H26N4O4
|
1
|
| 1 |
EC50 = 850 nM
|
|
|
|
CP0557087
|
N-(2-hydroxyethyl)-1-[6-[3-(trifluoromethyl)benzoyl]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H19F3N4O3
|
1
|
| 1 |
EC50 = 1008 nM
|
|
|
|
CP0465620
|
N-(2-hydroxyethyl)-1-[6-[3-(trifluoromethyl)anilino]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C22H20F3N5O2
|
1
|
| 1 |
EC50 = 1105 nM
|
|
|
|
CP0495719
|
1-[4-[3-fluoro-5-(trifluoromethyl)benzoyl]pyrimidin-2-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H18F4N4O3
|
1
|
| 1 |
EC50 = 1589 nM
|
|
|
|
CP0465608
|
1-[6-[3-fluoro-5-(trifluoromethyl)benzoyl]pyrimidin-4-yl]-N-(2-hydroxyethyl)-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C23H18F4N4O3
|
1
|
| 1 |
EC50 = 1693 nM
|
|
|
|
CP0533957
|
N-(2-hydroxyethyl)-1-[6-[3-(trifluoromethyl)phenoxy]pyrimidin-4-yl]-2,3-dihydroindole-4-carboxamide
Show/Hide
|
C22H19F3N4O3
|
1
|
| 1 |
EC50 = 2404 nM
|
|
|
|
CP0444098
|
(E)-1-(furan-2-yl)-5-phenylpent-2-en-1-one
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|
C15H14O2
|
1
|
| 1 |
IC50 = 630 nM
|
|
|
|
CP0558354
|
(E)-1,5-diphenylpent-2-en-1-one
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|
C17H16O
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0490660
|
(E)-5-phenyl-1-thiophen-2-ylpent-2-en-1-one
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|
C15H14OS
|
1
|
| 1 |
IC50 = 880 nM
|
|
|
|
CP0575624
|
(E)-5-phenyl-1-thiophen-3-ylpent-2-en-1-one
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|
C15H14OS
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0576628
|
(E)-5-phenyl-1-pyridin-3-ylpent-2-en-1-one
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|
C16H15NO
|
1
|
| 1 |
IC50 = 1010 nM
|
|
|
|
CP0490661
|
(E)-1-(2-methylpyrazol-3-yl)-5-phenylpent-2-en-1-one
Show/Hide
|
C15H16N2O
|
1
|
| 1 |
IC50 = 1080 nM
|
|
|
|
CP0490658
|
(E)-5-phenyl-1-(2-phenylphenyl)pent-2-en-1-one
Show/Hide
|
C23H20O
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
|
CP0573387
|
(E)-1-(3-methoxyphenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C18H18O2
|
1
|
| 1 |
IC50 = 1490 nM
|
|
|
|
CP0516886
|
(E)-1-(furan-3-yl)-5-phenylpent-2-en-1-one
Show/Hide
|
C15H14O2
|
1
|
| 1 |
IC50 = 1520 nM
|
|
|
|
CP0575621
|
(E)-5-(2-bromophenyl)-1-phenylpent-2-en-1-one
Show/Hide
|
C17H15BrO
|
1
|
| 1 |
IC50 = 1640 nM
|
|
|
|
CP0533081
|
(E)-1-(2-methoxyphenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C18H18O2
|
1
|
| 1 |
IC50 = 1720 nM
|
|
|
|
CP0577620
|
(E)-1-(2-fluorophenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C17H15FO
|
1
|
| 1 |
IC50 = 1760 nM
|
|
|
|
CP0490656
|
(E)-5-(4-bromophenyl)-1-phenylpent-2-en-1-one
Show/Hide
|
C17H15BrO
|
1
|
| 1 |
IC50 = 1810 nM
|
|
|
|
CP0577621
|
(E)-5-phenyl-1-pyridin-4-ylpent-2-en-1-one
Show/Hide
|
C16H15NO
|
1
|
| 1 |
IC50 = 1810 nM
|
|
|
|
CP0575040
|
(E)-5-phenyl-1-pyridin-2-ylpent-2-en-1-one
Show/Hide
|
C16H15NO
|
1
|
| 1 |
IC50 = 1820 nM
|
|
|
|
CP0444096
|
(E)-1-(3-fluorophenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C17H15FO
|
1
|
| 1 |
IC50 = 2370 nM
|
|
|
|
CP0534091
|
(E)-1-(3-methylphenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C18H18O
|
1
|
| 1 |
IC50 = 2570 nM
|
|
|
|
CP0575039
|
(E)-1-(2-methylphenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C18H18O
|
1
|
| 1 |
IC50 = 2630 nM
|
|
|
|
CP0558355
|
(E)-1-(2,6-dimethylphenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C19H20O
|
1
|
| 1 |
IC50 = 2820 nM
|
|
|
|
CP0490657
|
(E)-1-(4-methylphenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C18H18O
|
1
|
| 1 |
IC50 = 3020 nM
|
|
|
|
CP0573388
|
(E)-1-naphthalen-1-yl-5-phenylpent-2-en-1-one
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|
C21H18O
|
1
|
| 1 |
IC50 = 3290 nM
|
|
|
|
CP0533082
|
(E)-1-naphthalen-2-yl-5-phenylpent-2-en-1-one
Show/Hide
|
C21H18O
|
1
|
| 1 |
IC50 = 3540 nM
|
|
|
|
CP0574764
|
(E)-1-(4-methoxyphenyl)-5-phenylpent-2-en-1-one
Show/Hide
|
C18H18O2
|
1
|
| 1 |
IC50 = 3870 nM
|
|
|
|
CP0537593
|
(E)-1,7-diphenylhept-4-en-3-one
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|
C19H20O
|
1
|
| 1 |
IC50 = 5450 nM
|
|
|
|
CP0575623
|
(E)-5-phenyl-1-(4-phenylphenyl)pent-2-en-1-one
Show/Hide
|
C23H20O
|
1
|
| 1 |
IC50 = 7640 nM
|
|
|
|
CP0490659
|
(E)-5-phenyl-1-(3-phenylphenyl)pent-2-en-1-one
Show/Hide
|
C23H20O
|
1
|
| 1 |
IC50 = 8130 nM
|
|
|
