Brief Information of the Cell Line and Protein
Cell Line ID: CL000006 , HEK293
Synonyms
Hek293
HEK-293
HEK/293
HEK 293
HEK;293
293
293 HEK
293 Ad5
Graham 293
Graham-293
Human Embryonic Kidney 293
Category Transformed cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0045
Protein ID: PT02002 , Gamma-aminobutyric acid receptor subunit alpha-5
Gene Name GABRA5
Organism Homo sapiens, Human
Protein Classification Ion channel
Uniprot ID P31644
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000006  Protein ID: PT02002
 
Compound ID Compound Name Compound Formula
CP0551322
US8778932, 36
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C19H12FN3O2S
 1
1
IC50 = 100 nM
   TI
   LI
   LO
   TS
CP0379892
US8778932, 6
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C19H13N3O2S
 1
1
IC50 = 130 nM
   TI
   LI
   LO
   TS
CP0526532
US8778932, 21
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C19H12FN3O2S
 1
1
IC50 = 200 nM
   TI
   LI
   LO
   TS
CP0569564
US8778932, 9
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C20H11ClF3N3O2S
 1
1
IC50 = 250 nM
   TI
   LI
   LO
   TS
CP0412460
US8778932, 31
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C20H12F3N3O2S
 1
1
IC50 = 500 nM
   TI
   LI
   LO
   TS