(1S,2R,10S,11S,14S,15R,17S)-17-hydroxy-14-(2-hydroxyacetyl)-2-methyl-5-oxotetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadec-6-ene-15-carbaldehyde

(2R)-3-[[(8S,9S,10R,11S,13S,14S,17S)-17-acetyl-10,13-dimethyl-3-oxo-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-11-yl]amino]-2-aminopropanoic acid

4-(((6-((3-(2,6-dichlorophenyl)-5-isopropylisoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid

3-(((6-((5-cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid

4-(((6-((5-cyclopropyl-3-(2,6-dichlorophenyl)isoxazol-4-yl)methoxy)-2-(trifluoromethyl)pyridin-3-yl)(methyl)amino)methyl)benzoic acid

11BETA-HYDROXYPROGESTERONE

6-[5-(4-fluorophenyl)-3-methyl-1-(4,4,4-trifluorobutyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[1-(3,3-difluorobutyl)-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

8-chloro-6-[2-(4-fluoro-2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(4-fluoro-2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-8-methyl-4H-1,4-benzoxazin-3-one

[5-[(E)-(3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene)methyl]-1-[(2R)-1-morpholin-4-ylpropan-2-yl]benzimidazol-2-yl]cyanamide

6-[1-butyl-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

8-chloro-6-[4-(4-fluorophenyl)-2-methyl-5-oxo-1,2-dihydropyrrol-3-yl]-4H-1,4-benzoxazin-3-one

(S)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethyl)-1H-indol-7-yl)methanesulfonamide

6-[1-ethyl-4-(4-fluorophenyl)-2-methyl-5-oxo-2H-pyrrol-3-yl]-4H-1,4-benzoxazin-3-one

6-(2-phenyl-2H-imidazo[2,1-b][1,3,4]thiadiazin-3-yl)-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-3-methyl-1-(pyridin-3-ylmethyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[1-(2,2-difluoro-4-hydroxybutyl)-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[2-(4-fluoro-2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[4-(4-fluorophenyl)-2-methyl-5-oxo-1,2-dihydropyrrol-3-yl]-8-methyl-4H-1,4-benzoxazin-3-one

2',15'-dimethyl-5,5'-dioxo-(9'R)-spiro[tetrahydrofuran-2,14'-tetracyclo[8.7.0.02,7.011,15]heptadec-6'-ene]-9-yl ethanethioate

6-[1-(2,2-difluoro-3-hydroxypropyl)-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one

N-(3-(1-cyclopropyl-1-(4-fluorophenyl)ethyl)-1H-indol-7-yl)methanesulfonamide

6-[1-cyclopropyl-4-(4-fluorophenyl)-2-methyl-5-oxo-2H-pyrrol-3-yl]-4H-1,4-benzoxazin-3-one

6-(2-phenyl-2H-1,4-benzothiazin-3-yl)-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-1-(4-hydroxybutyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

8-fluoro-6-[2-(4-fluoro-2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(2-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-3-methyl-1-propylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

8-fluoro-6-[4-(4-fluorophenyl)-2-methyl-5-oxo-1,2-dihydropyrrol-3-yl]-4H-1,4-benzoxazin-3-one

6-[4-(4-fluorophenyl)-2-methyl-5-oxo-1,2-dihydropyrrol-3-yl]-4H-1,4-benzoxazin-3-one

6-[1-(3,3-difluoro-4-hydroxybutyl)-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[1-benzyl-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-1,3-dimethylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[4-(4-fluorophenyl)-2-methyl-5-oxo-2H-furan-3-yl]-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-1,3-dimethylpyrazol-4-yl]-8-methyl-4H-1,4-benzoxazin-3-one

6-[4-(4-fluorophenyl)-1,2-dimethyl-5-oxo-2H-pyrrol-3-yl]-4H-1,4-benzoxazin-3-one

6-[5-(2,4-difluorophenyl)-1,3-dimethylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

N-[2-[5-(4-fluorophenyl)-3-methyl-4-(3-oxo-4H-1,4-benzoxazin-6-yl)pyrazol-1-yl]ethyl]methanesulfonamide

6-[2-(4-fluorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[7-(4-fluorophenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl]-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-1-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

(R)-N-(3-(1-cyclopropyl-1-(2,4-difluorophenyl)ethyl)-1H-indol-7-yl)methanesulfonamide

6-[7-(3-fluorophenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl]-4H-1,4-benzoxazin-3-one

6-[2-(4-chlorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(2-chlorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(2-fluorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-1-(3-hydroxypropyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[4-(4-fluorophenyl)-5-oxo-2H-furan-3-yl]-4H-1,4-benzoxazin-3-one

6-(7-phenyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl)-4H-1,4-benzoxazin-3-one

6-[1-ethyl-5-(4-fluorophenyl)-3-methylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-3-methyl-1-(pyridin-4-ylmethyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one

3-[5-(4-fluorophenyl)-3-methyl-4-(3-oxo-4H-1,4-benzoxazin-6-yl)pyrazol-1-yl]propanenitrile

6-[2-fluoro-4-(4-fluorophenyl)-2-methyl-5-oxofuran-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(4-fluorophenyl)-5-(1,1,2,2,2-pentafluoroethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(4-methylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[7-(2-fluorophenyl)-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl]-4H-1,4-benzoxazin-3-one

6-[4-(2,4-difluorophenyl)-5-oxo-2H-furan-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(2-ethylphenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[4-(4-fluorophenyl)-5-methyl-1,2-oxazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[4-(4-fluoro-2-methylphenyl)-5-oxo-2H-furan-3-yl]-4H-1,4-benzoxazin-3-one

1-(4-fluorophenyl)-5-(3-oxo-4H-1,4-benzoxazin-6-yl)pyrazole-3-carbonitrile

6-[5-ethyl-2-(4-fluorophenyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(4-fluorophenyl)-5-methylpyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-(3-fluorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[4-(4-fluorophenyl)-2,2-dimethyl-5-oxofuran-3-yl]-4H-1,4-benzoxazin-3-one

6-[2-ethyl-4-(4-fluorophenyl)-5-oxo-2H-furan-3-yl]-4H-1,4-benzoxazin-3-one

6-(7-benzyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl)-4H-1,4-benzoxazin-3-one

6-[4-(4-fluorophenyl)-1-(2-hydroxyethyl)-2-methyl-5-oxo-2H-pyrrol-3-yl]-4H-1,4-benzoxazin-3-one

6-(7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl)-4H-1,4-benzoxazin-3-one

N-[3-(4-cyano-3-methoxyphenyl)-1-propan-2-ylindol-6-yl]methanesulfonamide

methyl (1R,2S,9R,10R,11S,14R,15S,17R)-2,15-dimethyl-5,5'-dioxospiro[18-oxapentacyclo[8.8.0.01,17.02,7.011,15]octadec-6-ene-14,2'-oxolane]-9-carboxylate

6-[2-(4-fluorophenyl)-4-(trifluoromethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-[5-(4-fluorophenyl)-3-methyl-1-(pyridin-2-ylmethyl)pyrazol-4-yl]-4H-1,4-benzoxazin-3-one

11BETA-AZIDOPROGESTERONE

6-[4-(4-fluorophenyl)-5-methyl-1H-pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

6-(7-propyl-7H-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl)-4H-1,4-benzoxazin-3-one

6-(5-methyl-2-phenylpyrazol-3-yl)-4H-1,4-benzoxazin-3-one

6-[2-(4-fluorophenyl)-5-(hydroxymethyl)pyrazol-3-yl]-4H-1,4-benzoxazin-3-one

N-[3-(4-cyano-3-fluorophenyl)-1-propan-2-ylindol-6-yl]methanesulfonamide

(S)-N-(1-sec-butyl-3-(4-cyanophenyl)-1H-indol-6-yl)methanesulfonamide

(R)-N-(1-sec-butyl-3-(4-cyanophenyl)-1H-indol-6-yl)methanesulfonamide

N-[3-(4-cyanophenyl)-1-ethylindol-6-yl]methanesulfonamide

3-[(4-methoxyphenyl)phenylmethyl]indole

N-[3-(4-cyano-3-methylphenyl)-1-propan-2-ylindol-6-yl]methanesulfonamide

N-[3-(4-cyanophenyl)-1-propan-2-ylindol-6-yl]methanesulfonamide

N-[3-(4-cyanophenyl)-1-methylindol-6-yl]methanesulfonamide

6-(2-methyl-5-phenyl-1H-imidazol-4-yl)-4H-1,4-benzoxazin-3-one

6-(7-methyl-7-phenyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazin-6-yl)-4H-1,4-benzoxazin-3-one

6-(2-methyl-5-phenyl-1,3-thiazol-4-yl)-4H-1,4-benzoxazin-3-one

6-[2-(4-fluorophenyl)-5-propan-2-ylpyrazol-3-yl]-4H-1,4-benzoxazin-3-one

N-[2-[5-(4-fluorophenyl)-3-methyl-4-(3-oxo-4H-1,4-benzoxazin-6-yl)pyrazol-1-yl]ethyl]acetamide

6-[5-(4-fluorophenyl)-3-methyl-1-phenylpyrazol-4-yl]-4H-1,4-benzoxazin-3-one

N-[(8S,9S,10R,11S,13S,14S,17S)-17-acetyl-10,13-dimethyl-3-oxo-1,2,6,7,8,9,11,12,14,15,16,17-dodecahydrocyclopenta[a]phenanthren-11-yl]-2-nitrobenzenesulfonamide

[5-[(E)-(3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene)methyl]-1-(4-methylpiperazin-1-yl)benzimidazol-2-yl]cyanamide

[1-[(7S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-5-[(E)-(3,7-difluoro-6H-benzo[c][1]benzoxepin-11-ylidene)methyl]benzimidazol-2-yl]cyanamide

(1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-hydroxyacetyl)-2,15-dimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-3,6-dien-5-one

[5-[(E)-(3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene)methyl]-1-[(2R)-1-morpholin-4-ylpropan-2-yl]benzimidazol-2-yl]urea

N-[3-[(1E)-1-(6H-benzo[c][1]benzoxepin-11-ylidene)ethyl]phenyl]methanesulfonamide

(1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dihydroxy-14-(2-hydroxyacetyl)-2,13,15-trimethyltetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-3,6-dien-5-one

[5-[(E)-(3,8-difluoro-6H-benzo[c][1]benzoxepin-11-ylidene)methyl]-1-[(2R)-1-morpholin-4-ylpropan-2-yl]benzimidazol-2-yl]cyanamide

N-[3-[(1E)-1-(6H-benzo[c][1]benzoxepin-11-ylidene)propyl]phenyl]methanesulfonamide

N-[3-(3-chlorophenyl)-1H-indol-7-yl]methanesulfonamide

N-[3-(2-tricyclo[9.4.0.03,8]pentadeca-1(15),3,5,7,11,13-hexaenylidenemethyl)phenyl]methanesulfonamide

N-[3-[(1Z)-1-(10-methoxy-6H-benzo[c][1]benzoxepin-11-ylidene)propyl]phenyl]methanesulfonamide

3-[(7R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl]-6-[(E)-(3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene)methyl]-1H-benzimidazol-2-one

N-(5-((3,7-difluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((7S,8aS)-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)cyanamide

N-(5-((3,7-difluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((R)-1-morpholinopropan-2-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)cyanamide

N-(5-((3,7-difluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((7R,8aR)-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)cyanamide

1-(5-((3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((7S,8aR)-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)urea

N-(5-((3,7-difluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((7R,8aS)-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-7-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)cyanamide

N-(5-((3,8-difluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((S)-1-morpholinopropan-2-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)cyanamide

N-(5-((3,7-difluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((S)-1-morpholinopropan-2-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)cyanamide

N-(5-((3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((S)-1-morpholinopropan-2-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)cyanamide

N-(5-((3-fluorodibenzo[b,e]oxepin-11(6H)-ylidene)methyl)-1-((3S,4S)-4-hydroxy-1-methylpyrrolidin-3-yl)-1H-benzo[d]imidazol-2(3H)-ylidene)cyanamide

5-[(E)-(3-fluoro-6H-benzo[c][1]benzoxepin-11-ylidene)methyl]-1,3-dihydrobenzimidazol-2-one

N-[3-(2-methoxyphenyl)-1H-indol-7-yl]methanesulfonamide

N-[3-(5-fluoro-2-methoxyphenyl)-5-methoxy-2-methyl-1H-indol-7-yl]methanesulfonamide

N-[5-fluoro-3-(4-fluoro-2-methoxyphenyl)-2-methyl-1H-indol-7-yl]methanesulfonamide

N-[3-(4-fluorophenyl)-1H-indol-7-yl]methanesulfonamide

(10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]-14-hydroxy-15-methyl-14-(prop-1-yn-1-yl)tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-1,6-dien-5-one

N-(1H-indol-7-yl)methanesulfonamide

N-[2-[[benzyl(methyl)amino]methyl]-3-(4-fluoro-2-methoxyphenyl)-5-propan-2-yl-1H-indol-7-yl]methanesulfonamide

2-[[benzyl(methyl)amino]methyl]-5-fluoro-3-(4-fluoro-2-methoxyphenyl)-1H-indol-7-amine

N-[2-[[benzyl(methyl)amino]methyl]-5-tert-butyl-3-(4-fluoro-2-methoxyphenyl)-1H-indol-7-yl]methanesulfonamide

N-(5-methoxy-2-methyl-3-phenyl-1H-indol-7-yl)methanesulfonamide

N-[3-(5-fluoro-2-methoxyphenyl)-2-phenyl-1H-indol-7-yl]methanesulfonamide

N-[2-benzyl-3-(4-fluoro-2-methoxyphenyl)-5-propan-2-yl-1H-indol-7-yl]methanesulfonamide

N-[3-(5-chloro-2-methoxyphenyl)-1H-indol-7-yl]methanesulfonamide

N-[3-(5-fluoro-2-methoxyphenyl)-1H-indol-7-yl]acetamide

N-(3-(1-cyclopropyl-1-phenylethyl)-1H-indol-7-yl)methanesulfonamide

N-(3-(1-cyclopropyl-1-p-tolylethyl)-1H-indol-7-yl)methanesulfonamide

N-(3-(3-phenylpentan-3-yl)-1H-indol-7-yl)methanesulfonamide

N-(3-(3-(4-chlorophenyl)pentan-3-yl)-1H-indol-7-yl)methanesulfonamide

N-(3-(3-(benzo[d]thiazol-6-yl)pentan-3-yl)-1H-indol-7-yl)methanesulfonamide

N-(3-(3-(4-hydroxyphenyl)pentan-3-yl)-1H-indol-7-yl)methanesulfonamide

N-(3-(3-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)pentan-3-yl)-1H-indol-7-yl)methanesulfonamide

N-(3-(3-(benzofuran-2-yl)pentan-3-yl)-1H-indol-7-yl)methanesulfonamide