| Compound ID |
Compound Name |
Compound Formula |
|
CP0078933
|
(-)-(1S,2S,3R,4R)-3-[(1S)-1-(Acetylamino)-2-ethylbutyl]-4-{[amino(imino)methyl]amino}-2-hydroxycyclopentanecarboxylic Acid
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|
C15H28N4O4
|
8
|
| 1 |
IC50 = 0.07 nM
|
|
|
| 2 |
IC50 = 0.3 nM
|
|
|
| 3 |
IC50 = 0.7 nM
|
|
|
| 4 |
IC50 = 0.8 nM
|
|
|
| 5 |
IC50 = 3.3 nM
|
|
|
| 6 |
IC50 = 3.6 nM
|
|
|
| 7 |
IC50 = 146 nM
|
|
|
| 8 |
IC50 = 225 nM
|
|
|
|
CP0386403
|
[(3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)cyclopenten-1-yl]phosphonic acid
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|
C14H27N4O4P
|
7
|
| 1 |
IC50 = 0.3 nM
|
|
|
| 2 |
IC50 = 2.3 nM
|
|
|
| 3 |
IC50 = 4.1 nM
|
|
|
| 4 |
IC50 = 73 nM
|
|
|
| 5 |
IC50 = 86 nM
|
|
|
| 6 |
IC50 = 2131 nM
|
|
|
| 7 |
IC50 > 83000 nM
|
|
|
|
CP0046477
|
(3R,4R,5S)-5-amino-4-acetamido-3-(pentan-3-yloxy)cyclohex-1-ene-1-carboxylic acid
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|
C14H24N2O4
|
8
|
| 1 |
IC50 = 0.4 nM
|
|
|
| 2 |
IC50 = 0.6 nM
|
|
|
| 3 |
IC50 = 0.9 nM
|
|
|
| 4 |
IC50 = 1 nM
|
|
|
| 5 |
IC50 = 26 nM
|
|
|
| 6 |
IC50 = 49 nM
|
|
|
| 7 |
IC50 = 4371 nM
|
|
|
| 8 |
IC50 > 83000 nM
|
|
|
|
CP0446358
|
[(1S,2S,3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)-2-hydroxycyclopentyl]-hexoxyphosphinic acid
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|
C20H41N4O5P
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0036726
|
(2R,3R,4S)-4-carbamimidamido-3-acetamido-2-[(1R,2R)-1,2,3-trihydroxypropyl]-3,4-dihydro-2H-pyran-6-carboxylic acid
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|
C12H20N4O7
|
8
|
| 1 |
IC50 = 0.6 nM
|
|
|
| 2 |
IC50 = 0.7 nM
|
|
|
| 3 |
IC50 = 1.7 nM
|
|
|
| 4 |
IC50 = 1.9 nM
|
|
|
| 5 |
IC50 = 4.2 nM
|
|
|
| 6 |
IC50 = 6 nM
|
|
|
| 7 |
IC50 = 45 nM
|
|
|
| 8 |
IC50 > 83000 nM
|
|
|
|
CP0447451
|
[(3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)cyclopenten-1-yl]-ethoxyphosphinic acid
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|
C16H31N4O4P
|
8
|
| 1 |
IC50 = 0.6 nM
|
|
|
| 2 |
IC50 = 0.9 nM
|
|
|
| 3 |
IC50 = 6.4 nM
|
|
|
| 4 |
IC50 = 7.3 nM
|
|
|
| 5 |
IC50 = 177 nM
|
|
|
| 6 |
IC50 = 187 nM
|
|
|
| 7 |
IC50 = 7481 nM
|
|
|
| 8 |
IC50 > 83000 nM
|
|
|
|
CP0553099
|
[(1S,2S,3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)-2-hydroxycyclopentyl]-ethoxyphosphinic acid
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|
C16H33N4O5P
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0474190
|
[(1S,2S,3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)-2-hydroxycyclopentyl]phosphonic acid
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|
C14H29N4O5P
|
8
|
| 1 |
IC50 = 0.9 nM
|
|
|
| 2 |
IC50 = 1.9 nM
|
|
|
| 3 |
IC50 = 3.1 nM
|
|
|
| 4 |
IC50 = 5.2 nM
|
|
|
| 5 |
IC50 = 627 nM
|
|
|
| 6 |
IC50 = 705 nM
|
|
|
| 7 |
IC50 = 2831 nM
|
|
|
| 8 |
IC50 > 83000 nM
|
|
|
|
CP0571165
|
[(1R,3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)cyclopentyl]-ethoxyphosphinic acid
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|
C16H33N4O4P
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0409697
|
[(3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)cyclopenten-1-yl]-hexoxyphosphinic acid
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|
C20H39N4O4P
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0451988
|
[(1R,3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)cyclopentyl]-hexoxyphosphinic acid
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|
C20H41N4O4P
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0549179
|
[(1R,3S,4R)-3-[(1S)-1-acetamido-2-ethylbutyl]-4-(diaminomethylideneamino)cyclopentyl]phosphonic acid
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|
C14H29N4O4P
|
1
|
| 1 |
IC50 = 2.9 nM
|
|
|
