| Compound ID |
Compound Name |
Compound Formula |
|
CP0330041
|
N-cyclopropyl-4-(2-pyridin-2-ylpyrrolidin-1-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
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|
C20H21N5O
|
1
|
| 1 |
EC50 = 1.995 nM
|
|
|
|
CP0547521
|
N-ethyl-4-(2-phenylpyrrolidin-1-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
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|
C20H22N4O
|
1
|
| 1 |
EC50 = 1.995 nM
|
|
|
|
CP0349171
|
17-(methylamino)-8,11,14-trioxa-1,16,19,22-tetrazatetracyclo[13.5.2.13,7.018,21]tricosa-3(23),4,6,15,17,21-hexaen-20-one
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|
C17H19N5O4
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0229824
|
4-(4-chloro-2-fluoroanilino)-6,7-dimethoxy-N-methylquinoline-3-carboxamide
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|
C19H17ClFN3O3
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0354226
|
17-(methylamino)-8,14-dioxa-1,16,19,22-tetrazatetracyclo[13.5.2.13,7.018,21]tricosa-3(23),4,6,15,17,21-hexaen-20-one
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|
C18H21N5O3
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0390117
|
N-(oxetan-3-yl)-4-(2-pyridin-2-ylpyrrolidin-1-yl)-1H-pyrrolo[2,3-b]pyridine-2-carboxamide
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|
C20H21N5O2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0274216
|
4-N-cyclopropyl-6-(2,3-dichlorophenyl)pyrimidine-2,4-diamine
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|
C13H12Cl2N4
|
2
|
| 1 |
EC50 = 10 nM
|
|
|
| 2 |
EC50 = 125.89 nM
|
|
|
|
CP0330038
|
4-(2-phenylpyrrolidin-1-yl)-1H-pyrrolo[2,3-b]pyridine
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|
C17H17N3
|
1
|
| 1 |
EC50 = 63.1 nM
|
|
|
|
CP0143330
|
4-[4-[2-(dimethylamino)ethyl]phenyl]quinazolin-2-amine
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|
C18H20N4
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0390118
|
4-(2-pyridin-3-ylpyrrolidin-1-yl)-1H-pyrazolo[3,4-b]pyridine
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|
C15H15N5
|
1
|
| 1 |
EC50 = 251.19 nM
|
|
|
|
CP0229823
|
4-(4-chloro-2-fluoroanilino)-6,7-dimethoxy-N,N-dimethylquinoline-3-carboxamide
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|
C20H19ClFN3O3
|
1
|
| 1 |
EC50 = 950 nM
|
|
|
|
CP0354227
|
9-benzyl-2-(2-methoxyethoxy)-6-(methylamino)-7H-purin-8-one
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|
C16H19N5O3
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0229821
|
3-[(1S)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-ylpyrazol-4-yl)pyridin-2-amine
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|
C21H22Cl2FN5O
|
1
|
| 1 |
EC50 = 3600 nM
|
|
|