| Compound ID |
Compound Name |
Compound Formula |
|
CP0539851
|
US8802721, 1
Show/Hide
|
C18H9ClF5NOS
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0535639
|
US8802721, 3
Show/Hide
|
C20H15F2NO3S
|
1
|
| 1 |
IC50 = 6.4 nM
|
|
|
|
CP0533824
|
N-[4-[2-chloro-5-(trifluoromethyl)phenyl]phenyl]-2,6-difluorobenzamide
Show/Hide
|
C20H11ClF5NO
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0003531
|
2,6-difluoro-N-[4-[2-methyl-3-(4-methyl-5-oxo-1,3,4-oxadiazol-2-yl)phenyl]phenyl]benzamide
Show/Hide
|
C23H17F2N3O3
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0539711
|
US8802721, 2
Show/Hide
|
C18H12ClF3N2OS
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0565081
|
2-chloro-6-fluoro-N-[4-[2-methyl-3-(4-methyl-5-oxo-1,3,4-oxadiazol-2-yl)phenyl]phenyl]benzamide
Show/Hide
|
C23H17ClFN3O3
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0529364
|
US8802721, 117
Show/Hide
|
C18H10F5NOS
|
1
|
| 1 |
IC50 = 16.5 nM
|
|
|
|
CP0570245
|
N-[5-[5-(5,5-dimethyl-4-oxo-1,2-oxazol-3-yl)-2-ethylphenyl]pyrazin-2-yl]-2,6-difluorobenzamide
Show/Hide
|
C24H20F2N4O3
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0451107
|
2,6- Difluoro-N-(2′- methyl-5′-(4-methyl- 5-oxo-4,5-dihydro- 1,3,4-oxadiazol-2-yl)- [1,1′-biphenyl]-4- yl)benzamide
Show/Hide
|
C23H17F2N3O3
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0543909
|
N-[5-[5-(5,5-dimethyl-4-oxo-1,2-oxazol-3-yl)-2-methylphenyl]pyrazin-2-yl]-2,6-difluorobenzamide
Show/Hide
|
C23H18F2N4O3
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0571529
|
N-[5-[5-(5,5-dimethyl-4-oxo-1,2-oxazol-3-yl)-2-methoxyphenyl]pyrazin-2-yl]-2,6-difluorobenzamide
Show/Hide
|
C23H18F2N4O4
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0418566
|
N-[5-[3-(5,5-dimethyl-4-oxo-1,2-oxazol-3-yl)-2-methylphenyl]pyrazin-2-yl]-2,6-difluorobenzamide
Show/Hide
|
C23H18F2N4O3
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0551028
|
US8802721, 4
Show/Hide
|
C20H18N2O3S
|
1
|
| 1 |
IC50 = 58.5 nM
|
|
|
|
CP0533823
|
2,6- Difluoro-N-(5-(2- methyl-5-(4- methyl-5-oxo-4,5- dihydro-1,3,4- oxadiazol-2- yl)phenyl)pyrazin- 2-yl)benzamide
Show/Hide
|
C21H15F2N5O3
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0557778
|
2- Chloro-N-(5-(5-(5,5- dimethyl-4-oxo-4,5- dihydroisoxazol-3- yl)-2-methyl phenyl)pyrazin-2-yl)- 6-fluorobenzamide
Show/Hide
|
C23H18ClFN4O3
|
1
|
| 1 |
IC50 = 64.8 nM
|
|
|
|
CP0565080
|
N-(5′- (5,5-Dimethyl-4-oxo- 4,5-dihydroisoxazol- 3-yl)-2′-methyl-[1,1′- biphenyl]-4-yl-2,6- difluorobenzamide
Show/Hide
|
C25H20F2N2O3
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0557779
|
N-(5′- (4-Ethyl-5-oxo-4,5- dihydro-1,3,4- oxadiazol-2-yl)-2′- methyl-[1,1′- biphenyl]-4-yl)-2,6- difluorobenzamide
Show/Hide
|
C24H19F2N3O3
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0443018
|
US8802721, 120
Show/Hide
|
C20H15F2NO3S
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0559821
|
N-(5-(5- (5,5-dimethyl-4-oxo- 4,5-dihydroisoxazol-3- yl)-2- methylphenyl)pyrazin- 2-yl)-3,5- difluoroisonicotinamide
Show/Hide
|
C22H17F2N5O3
|
1
|
| 1 |
IC50 = 94.4 nM
|
|
|
|
CP0442352
|
US8802721, 119
Show/Hide
|
C21H14F2N2O2S
|
1
|
| 1 |
IC50 = 94.8 nM
|
|
|
|
CP0443016
|
US8802721, 118
Show/Hide
|
C20H15F2NO3S
|
1
|
| 1 |
IC50 = 103.6 nM
|
|
|
|
CP0569713
|
US10292981, Example 121
Show/Hide
|
C23H18F2N4O3
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0539712
|
US8802721, 121
Show/Hide
|
C20H12F2N2O2S
|
1
|
| 1 |
IC50 = 164.4 nM
|
|
|
|
CP0533844
|
US10292981, Example 78
Show/Hide
|
C23H19ClN4O3
|
1
|
| 1 |
IC50 = 171 nM
|
|
|
|
CP0571530
|
N-(5-(5- (5,5-Dimethyl-4-oxo- 4,5-dihydroisoxazol- 3-yl)-2- methylphenyl)pyridin- 2-yl)-2,6- difluorobenzamide
Show/Hide
|
C24H19F2N3O3
|
1
|
| 1 |
IC50 = 178 nM
|
|
|
|
CP0570373
|
2,6-difluoro-N-[4-[2-methyl-5-(2-oxo-3H-1,3,4-oxadiazol-5-yl)phenyl]phenyl]benzamide
Show/Hide
|
C22H15F2N3O3
|
1
|
| 1 |
IC50 = 227 nM
|
|
|
|
CP0485615
|
N-(5- (5,5-Dimethyl-4,5- dihydroisoxazol-3- yl)-2- methylphenyl)pyrazin- 2-yl)-2,6- difluorobenzamide
Show/Hide
|
C23H20F2N4O2
|
1
|
| 1 |
IC50 = 328 nM
|
|
|
