Compound ID |
Compound Name |
Compound Formula |
CP0125809
|
US9458171, 392
Show/Hide
|
C29H27F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0136114
|
US9458171, 387
Show/Hide
|
C29H29F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0202748
|
US9458171, 95
Show/Hide
|
C27H25F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384347
|
4-[(3R)-3-(4-fluorophenyl)sulfonyl-3-[4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)phenyl]pyrrolidine-1-carbonyl]-4-methylcyclohexane-1-carboxylic acid
Show/Hide
|
C28H27F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384348
|
4-[(3R)-3-(4-fluorophenyl)sulfonyl-3-[4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)phenyl]pyrrolidine-1-carbonyl]-4-(methoxymethyl)cyclohexane-1-carboxylic acid
Show/Hide
|
C29H29F8NO6S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384357
|
US9458171, 499
Show/Hide
|
C27H27F8NO5S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384652
|
US9458171, 103
Show/Hide
|
C27H26F8N2O4S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384653
|
US9458171, 494
Show/Hide
|
C26H25F8NO5S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384656
|
US9458171, 402
Show/Hide
|
C28H25F8NO6S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384659
|
US9458171, 502
Show/Hide
|
C25H23F8NO6S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384660
|
US9458171, 382
Show/Hide
|
C28H27F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384661
|
4-[(3R)-3-(4-fluorophenyl)sulfonyl-3-[4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)phenyl]pyrrolidine-1-carbonyl]-4-methylcyclohexane-1-carboxylic acid
Show/Hide
|
C28H27F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384662
|
US9458171, 101
Show/Hide
|
C27H25F8NO6S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0384663
|
US9458171, 485
Show/Hide
|
C25H23F8NO5S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0416603
|
US9458171, 399
Show/Hide
|
C27H23F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0416604
|
US9458171, 403
Show/Hide
|
C28H25F8NO6S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0416605
|
US9458171, 405
Show/Hide
|
C28H25F8N3O5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0416606
|
US9458171, 411
Show/Hide
|
C28H27F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0416621
|
US9458171, 397
Show/Hide
|
C28H25F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0416623
|
US9458171, 489
Show/Hide
|
C24H21F8NO5S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0416630
|
US9458171, 393
Show/Hide
|
C30H31F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0416632
|
US9458171, 396
Show/Hide
|
C29H29F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0434779
|
US9458171, 404
Show/Hide
|
C27H23F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0434781
|
US9458171, 504
Show/Hide
|
C26H25F8NO6S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0440422
|
US9458171, 533
Show/Hide
|
C27H27F8NO5S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0440423
|
US9458171, 400
Show/Hide
|
C27H23F8NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0440424
|
4-[(3R)-3-(4-fluorophenyl)sulfonyl-3-[4-(1,1,1,2,3,3,3-heptafluoropropan-2-yl)phenyl]pyrrolidine-1-carbonyl]-4-methoxycyclohexane-1-carboxylic acid
Show/Hide
|
C28H27F8NO6S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0440425
|
US9458171, 386
Show/Hide
|
C27H24F9NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0478420
|
US9458171, 385
Show/Hide
|
C27H24F9NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0478422
|
US9458171, 514
Show/Hide
|
C27H27F8NO4S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0535831
|
US9458171, 517
Show/Hide
|
C26H25F8NO4S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0535853
|
US9458171, 526
Show/Hide
|
C26H25F8NO6S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0548402
|
US9458171, 383
Show/Hide
|
C27H24F9NO5S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0553126
|
US9458171, 519
Show/Hide
|
C25H22F9NO5S2
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0867529
|
US9458171, 401
Show/Hide
|
C27H25F8N5O3S
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0311844
|
US11078186, Example 119
Show/Hide
|
C29H28F7N3O3
|
1
|
1 |
EC50 > 40000 nM
|
|
|
CP0408973
|
1,1,1,3,3,3-hexafluoro-2-[4-(4-fluorophenyl)sulfonyl-2,3-dihydro-1,4-benzothiazin-7-yl]propan-2-ol
Show/Hide
|
C17H12F7NO3S2
|
2
|
1 |
EC50 > 2000 nM
|
|
|
2 |
EC50 > 4000 nM
|
|
|
CP0904554
|
cis-3-({(5R)-5-[(7-Fluoro-1,1-dimethyl-2,3-dihydro-1H-inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5H)-yl}carbonyl)cyclobutyl]acetic Acid
Show/Hide
|
C28H32FN3O5
|
1
|
1 |
IC50 >= 30000 nM
|
|
|