Brief Information of the Cell Line and Protein
Cell Line ID: CL000001 , Jurkat
Synonyms
JURKAT
JM
JM-Jurkat
Jurkat-FHCRC
Jurkat FHCRC
FHCRC-11
FHCRC subclone 11
FCCH1024
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0065
Protein ID: PT01875 , cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
Gene Name PDE10A
Organism Homo sapiens, Human
Protein Classification Enzyme
Uniprot ID Q9Y233
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000001  Protein ID: PT01875
 
Compound ID Compound Name Compound Formula
CP0451477
US9464076, 54
   Show/Hide
C23H21N3O3S
 1
1
IC50 = 0.054 nM
   TI
   LI
   LO
   TS
CP0465862
US9464076, 58
   Show/Hide
C31H35N3O4S
 1
1
IC50 = 0.085 nM
   TI
   LI
   LO
   TS
CP0535678
US9464076, 101
   Show/Hide
C27H25N3O5S
 1
1
IC50 = 0.11 nM
   TI
   LI
   LO
   TS
CP0565324
US9464076, 93
   Show/Hide
C24H20N2O5S
 1
1
IC50 = 0.11 nM
   TI
   LI
   LO
   TS
CP0565328
US9464076, 99
   Show/Hide
C27H24FN3O4S
 1
1
IC50 = 0.11 nM
   TI
   LI
   LO
   TS
CP0475013
US9464076, 113
   Show/Hide
C24H22N2O4S
 1
1
IC50 = 0.12 nM
   TI
   LI
   LO
   TS
CP0567694
US9464076, 98
   Show/Hide
C27H25N3O4S
 1
1
IC50 = 0.21 nM
   TI
   LI
   LO
   TS
CP0104858
US9464076, 109
   Show/Hide
C25H24N2O5S2
 1
1
IC50 = 0.23 nM
   TI
   LI
   LO
   TS
CP0268614
US9464076, 38
   Show/Hide
C28H29N3O4S
 1
1
IC50 = 0.23 nM
   TI
   LI
   LO
   TS
CP0567693
US9464076, 97
   Show/Hide
C26H25N3O4S
 1
1
IC50 = 0.26 nM
   TI
   LI
   LO
   TS
CP0516370
US9464076, 35
   Show/Hide
C28H29N3O4S
 1
1
IC50 = 0.29 nM
   TI
   LI
   LO
   TS
CP0489598
US9464076, 59
   Show/Hide
C30H33N3O4S
 1
1
IC50 = 0.31 nM
   TI
   LI
   LO
   TS
CP0565326
US9464076, 96
   Show/Hide
C29H30N4O4S
 1
1
IC50 = 0.31 nM
   TI
   LI
   LO
   TS
CP0483252
US9464076, 36
   Show/Hide
C29H31N3O4S
 1
1
IC50 = 0.35 nM
   TI
   LI
   LO
   TS
CP0519230
US9464076, 65
   Show/Hide
C27H27N3O4S
 1
1
IC50 = 0.39 nM
   TI
   LI
   LO
   TS
CP0576963
US9464076, 100
   Show/Hide
C27H23F2N3O4S
 1
1
IC50 = 0.42 nM
   TI
   LI
   LO
   TS
CP0519229
US9464076, 46
   Show/Hide
C29H30FN3O3S
 1
1
IC50 = 0.44 nM
   TI
   LI
   LO
   TS
CP0535673
US9464076, 55
   Show/Hide
C25H25N3O3S
 1
1
IC50 = 0.45 nM
   TI
   LI
   LO
   TS
CP0471290
US9464076, 18
   Show/Hide
C26H26N2O3S
 1
1
IC50 = 0.47 nM
   TI
   LI
   LO
   TS
CP0483293
US9464076, 95
   Show/Hide
C28H27N3O5S
 1
1
IC50 = 0.48 nM
   TI
   LI
   LO
   TS
CP0465861
US9464076, 47
   Show/Hide
C27H27N3O4S
 1
1
IC50 = 0.49 nM
   TI
   LI
   LO
   TS
CP0483254
US9464076, 45
   Show/Hide
C28H28FN3O3S
 1
1
IC50 = 0.5 nM
   TI
   LI
   LO
   TS
CP0535670
US9464076, 37
   Show/Hide
C29H31N3O4S
 1
1
IC50 = 0.5 nM
   TI
   LI
   LO
   TS
CP0444981
US9464076, 76
   Show/Hide
C25H24N2O4S
 1
1
IC50 = 0.53 nM
   TI
   LI
   LO
   TS
CP0497605
US9464076, 72
   Show/Hide
C26H26N2O5S
 1
1
IC50 = 0.54 nM
   TI
   LI
   LO
   TS
CP0190119
US9464076, 87
   Show/Hide
C24H23N2O7PS
 1
1
IC50 = 0.6 nM
   TI
   LI
   LO
   TS
CP0575945
US9464076, 21
   Show/Hide
C27H26N2O3S
 1
1
IC50 = 0.67 nM
   TI
   LI
   LO
   TS
CP0483292
US9464076, 91
   Show/Hide
C27H27N3O6S
 1
1
IC50 = 0.74 nM
   TI
   LI
   LO
   TS
CP0471286
US9464076, 71
   Show/Hide
C27H28N2O5S
 1
1
IC50 = 0.75 nM
   TI
   LI
   LO
   TS
CP0576961
US9464076, 64
   Show/Hide
C28H29N3O4S
 1
1
IC50 = 0.76 nM
   TI
   LI
   LO
   TS
CP0488592
US9464076, 125
   Show/Hide
C29H32N4O3S
 1
1
IC50 = 0.8 nM
   TI
   LI
   LO
   TS
CP0576957
US9464076, 48
   Show/Hide
C28H27F2N3O3S
 1
1
IC50 = 0.85 nM
   TI
   LI
   LO
   TS
CP0535676
US9464076, 83
   Show/Hide
C26H24N2O5S
 1
1
IC50 = 0.86 nM
   TI
   LI
   LO
   TS
CP0405879
US9464076, 115
   Show/Hide
C27H25N3O5S
 1
1
IC50 = 0.89 nM
   TI
   LI
   LO
   TS
CP0500943
US9464076, 14
   Show/Hide
C24H20N2O4S
 1
1
IC50 = 0.89 nM
   TI
   LI
   LO
   TS
CP0497604
US9464076, 33
   Show/Hide
C25H24N2O4S
 1
1
IC50 = 0.9 nM
   TI
   LI
   LO
   TS
CP0517233
US9464076, 75
   Show/Hide
C25H22N2O4S
 1
1
IC50 = 0.91 nM
   TI
   LI
   LO
   TS
CP0465860
US9464076, 42
   Show/Hide
C29H31N3O4S
 1
1
IC50 = 0.92 nM
   TI
   LI
   LO
   TS
CP0556316
US9464076, 19
   Show/Hide
C26H24N2O3S
 1
1
IC50 = 0.92 nM
   TI
   LI
   LO
   TS
CP0405876
US9464076, 34
   Show/Hide
C27H29N3O4S
 1
1
IC50 = 0.94 nM
   TI
   LI
   LO
   TS
CP0493168
US9464076, 22
   Show/Hide
C27H28N2O3S
 1
1
IC50 = 1 nM
   TI
   LI
   LO
   TS
CP0444982
US9464076, 85
   Show/Hide
C26H25N3O5S
 1
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0465835
US9464076, 63
   Show/Hide
C28H29N3O4S
 1
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0483255
US9464076, 56
   Show/Hide
C27H27N3O4S
 1
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0567692
US9464076, 86
   Show/Hide
C27H27N3O5S
 1
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0576958
US9464076, 49
   Show/Hide
C23H20N2O3S
 1
1
IC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0535674
US9464076, 60
   Show/Hide
C28H28FN3O3S
 1
1
IC50 = 1.2 nM
   TI
   LI
   LO
   TS
CP0535677
US9464076, 94
   Show/Hide
C28H28N4O4S
 1
1
IC50 = 1.2 nM
   TI
   LI
   LO
   TS
CP0576962
US9464076, 66
   Show/Hide
C28H29N3O4S
 1
1
IC50 = 1.2 nM
   TI
   LI
   LO
   TS
CP0577345
US9464076, 52
   Show/Hide
C27H25N3O4S
 1
1
IC50 = 1.2 nM
   TI
   LI
   LO
   TS
CP0576960
US9464076, 61
   Show/Hide
C28H29N3O4S
 1
1
IC50 = 1.3 nM
   TI
   LI
   LO
   TS
CP0553707
US9464076, 51
   Show/Hide
C28H27N3O4S
 1
1
IC50 = 1.5 nM
   TI
   LI
   LO
   TS
CP0400481
US9464076, 108
   Show/Hide
C24H22N2O3S
 1
1
IC50 = 1.6 nM
   TI
   LI
   LO
   TS
CP0483257
US9464076, 70
   Show/Hide
C26H26N2O4S
 1
1
IC50 = 1.6 nM
   TI
   LI
   LO
   TS
CP0575942
US9464076, 1
   Show/Hide
C23H18N2O3S
 1
1
IC50 = 1.6 nM
   TI
   LI
   LO
   TS
CP0576959
US9464076, 57
   Show/Hide
C28H30N4O3S
 1
1
IC50 = 1.6 nM
   TI
   LI
   LO
   TS
CP0286054
US9464076, 26
   Show/Hide
C26H26N2O4S
 1
1
IC50 = 1.8 nM
   TI
   LI
   LO
   TS
CP0535675
US9464076, 62
   Show/Hide
C26H27N3O3S
 1
1
IC50 = 1.8 nM
   TI
   LI
   LO
   TS
CP0451482
US9464076, 73
   Show/Hide
C25H22F2N2O4S
 1
1
IC50 = 2 nM
   TI
   LI
   LO
   TS
CP0489594
US9464076, 13
   Show/Hide
C25H22N2O4S
 1
1
IC50 = 2 nM
   TI
   LI
   LO
   TS
CP0451353
US9464076, 114
   Show/Hide
C23H20N2O4S
 1
1
IC50 = 2.1 nM
   TI
   LI
   LO
   TS
CP0483253
US9464076, 44
   Show/Hide
C28H29N3O4S
 1
1
IC50 = 2.1 nM
   TI
   LI
   LO
   TS
CP0577344
US9464076, 11
   Show/Hide
C24H20N2O3S
 1
1
IC50 = 2.2 nM
   TI
   LI
   LO
   TS
CP0471289
US9464076, 15
   Show/Hide
C27H25N3O4S
 1
1
IC50 = 2.3 nM
   TI
   LI
   LO
   TS
CP0265225
US9464076, 2
   Show/Hide
C26H24N2O4S
 1
1
IC50 = 2.6 nM
   TI
   LI
   LO
   TS
CP0535668
US9464076, 17
   Show/Hide
C26H26N2O3S
 1
1
IC50 = 2.6 nM
   TI
   LI
   LO
   TS
CP0535671
US9464076, 50
   Show/Hide
C28H27N3O5S
 1
1
IC50 = 2.6 nM
   TI
   LI
   LO
   TS
CP0405880
US9464076, 124
   Show/Hide
C28H30N4O3S
 1
1
IC50 = 2.9 nM
   TI
   LI
   LO
   TS
CP0405877
US9464076, 74
   Show/Hide
C26H26N2O4S
 1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
CP0576956
US9464076, 29
   Show/Hide
C27H28N2O4S
 1
1
IC50 = 3 nM
   TI
   LI
   LO
   TS
CP0535669
US9464076, 25
   Show/Hide
C28H28N2O3S
 1
1
IC50 = 4 nM
   TI
   LI
   LO
   TS
CP0490127
US9464076, 12
   Show/Hide
C24H20N2O4S
 1
1
IC50 = 4.4 nM
   TI
   LI
   LO
   TS
CP0535667
US9464076, 16
   Show/Hide
C25H24N2O3S
 1
1
IC50 = 4.8 nM
   TI
   LI
   LO
   TS
CP0575943
US9464076, 7
   Show/Hide
C27H26N2O4S
 1
1
IC50 = 5 nM
   TI
   LI
   LO
   TS
CP0517238
US9464076, 43
   Show/Hide
C28H29N3O3S
 1
1
IC50 = 6.2 nM
   TI
   LI
   LO
   TS
CP0483291
US9464076, 84
   Show/Hide
C29H31N3O5S
 1
1
IC50 = 7.1 nM
   TI
   LI
   LO
   TS
CP0575944
US9464076, 9
   Show/Hide
C26H26N2O4S
 1
1
IC50 = 7.8 nM
   TI
   LI
   LO
   TS
CP0493169
US9464076, 32
   Show/Hide
C27H28N2O4S
 1
1
IC50 = 9.1 nM
   TI
   LI
   LO
   TS
CP0405875
US9464076, 20
   Show/Hide
C27H28N2O3S
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0526119
US9464076, 23
   Show/Hide
C27H28N2O3S
 1
1
IC50 = 10 nM
   TI
   LI
   LO
   TS
CP0575946
US9464076, 30
   Show/Hide
C28H30N2O4S
 1
1
IC50 = 11 nM
   TI
   LI
   LO
   TS
CP0138175
US9464076, 8
   Show/Hide
C25H22N2O4S
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0405878
US9464076, 92
   Show/Hide
C25H22N2O5S
 1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS
CP0471285
US9464076, 31
   Show/Hide
C28H30N2O4S
 1
1
IC50 = 16 nM
   TI
   LI
   LO
   TS
CP0535672
US9464076, 53
   Show/Hide
C23H19ClN2O3S
 1
1
IC50 = 18 nM
   TI
   LI
   LO
   TS
CP0535666
US9464076, 10
   Show/Hide
C27H26N2O4S
 1
1
IC50 = 20 nM
   TI
   LI
   LO
   TS
CP0576955
US9464076, 24
   Show/Hide
C28H30N2O3S
 1
1
IC50 = 25 nM
   TI
   LI
   LO
   TS