| Compound ID |
Compound Name |
Compound Formula |
|
CP0076784
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]-3-methylphenyl]indazole-3-carboxamide
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|
C34H38N8O4
|
1
|
| 1 |
EC50 = 28 nM
|
|
|
|
CP0076786
|
N-[3-chloro-4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]phenyl]-1-[1-(3-cyano-3-methylbutanoyl)piperidin-4-yl]-5-fluoroindazole-3-carboxamide
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|
C34H32ClFN8O4
|
1
|
| 1 |
EC50 = 41 nM
|
|
|
|
CP0201458
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[3-methyl-4-(pyrazolo[1,5-a]pyridine-3-carbonylamino)phenyl]indazole-3-carboxamide
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|
C33H36N8O3
|
1
|
| 1 |
EC50 = 42 nM
|
|
|
|
CP0363721
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[3-chloro-4-(pyrazolo[1,5-a]pyridine-3-carbonylamino)phenyl]indazole-3-carboxamide
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|
C32H33ClN8O3
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0157559
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[3-chloro-4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]phenyl]-5-fluoroindazole-3-carboxamide
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|
C33H34ClFN8O4
|
1
|
| 1 |
EC50 = 56 nM
|
|
|
|
CP0076785
|
1-[1-(3-cyano-3-methylbutanoyl)piperidin-4-yl]-N-[3-methyl-4-(pyrazolo[1,5-a]pyridine-3-carbonylamino)phenyl]indazole-3-carboxamide
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|
C34H34N8O3
|
1
|
| 1 |
EC50 = 88 nM
|
|
|
|
CP0457470
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[4-(4,5-dimethyl-6-oxo-1H-pyridazin-3-yl)-3-ethylphenyl]indazole-3-carboxamide
Show/Hide
|
C32H39N7O3
|
1
|
| 1 |
EC50 = 420 nM
|
|
|
|
CP0201463
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[4-(pyrazolo[1,5-a]pyridine-3-carbonylamino)phenyl]indazole-3-carboxamide
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|
C32H34N8O3
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0426300
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[3-ethyl-4-(4-methyl-6-oxo-1H-pyridazin-3-yl)phenyl]indazole-3-carboxamide
Show/Hide
|
C31H37N7O3
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
|
CP0224675
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[3-ethyl-4-(5-methyl-6-oxo-1H-pyridazin-3-yl)phenyl]indazole-3-carboxamide
Show/Hide
|
C31H37N7O3
|
1
|
| 1 |
EC50 = 2700 nM
|
|
|
|
CP0457471
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[3-chloro-4-(4-methyl-6-oxo-1H-pyridazin-3-yl)phenyl]indazole-3-carboxamide
Show/Hide
|
C29H32ClN7O3
|
1
|
| 1 |
EC50 = 4050 nM
|
|
|
|
CP0076783
|
1-[1-(tert-butylcarbamoyl)piperidin-4-yl]-N-[3-chloro-4-(6-oxo-1H-pyridazin-3-yl)phenyl]indazole-3-carboxamide
Show/Hide
|
C28H30ClN7O3
|
1
|
| 1 |
EC50 = 5700 nM
|
|
|
|
CP0201461
|
1-[[1-(tert-butylcarbamoyl)azetidin-3-yl]methyl]-N-[3-chloro-4-(6-oxo-1H-pyridazin-3-yl)phenyl]indazole-3-carboxamide
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|
C27H28ClN7O3
|
1
|
| 1 |
EC50 = 7900 nM
|
|
|
|
CP0157558
|
N-[4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]-3-methylphenyl]-1-methylindazole-3-carboxamide
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|
C25H22N6O3
|
1
|
| 1 |
EC50 > 20000 nM
|
|
|
|
CP0093554
|
BIIB-057
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|
C19H23N9O
|
1
|
| 1 |
IC50 = 1805 nM
|
|
|
|
CP0658097
|
5-(1H-indol-7-ylamino)-3-((1R,2S)-2-aminocyclohexylamino)-1,2,4-triazine-6-carboxamide
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|
C18H22N8O
|
1
|
| 1 |
IC50 = 2526 nM
|
|
|
