Brief Information of the Compound and Protein
Compound Name
1-(2-methoxy-5-methylphenyl)-N-(2-methylquinolin-5-yl)sulfonyl-2-(6-propan-2-yloxypyridin-2-yl)cyclopropane-1-carboxamide
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PubChem ID
CID: 168270037
Canonical SMILES
COc1ccc(C)cc1C1(CC1c1cccc(OC(C)C)n1)C(=O)NS(=O)(=O)c1cccc2nc(C)ccc12
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Compound Formula C30H31N3O5S
Compound Structure
Protein Name
Cystic fibrosis transmembrane conductance regulator
Protein Classification
Ion channel
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Other ion channel
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Chloride channel
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Cystic fibrosis transmembrane conductance regulator
Uniprot ID
P13569
Gene Name
CFTR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000805 HBE1 Homo sapiens (Human)  1
1
EC50 = 0.9 nM
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