Brief Information of the Compound and Protein
Compound Name
2-[(2-amino-3-methylquinolin-7-yl)methyl]-N-(3-fluoropyridin-2-yl)-N-methylpyrazole-3-carboxamide
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PubChem ID
CID: 168289460
Canonical SMILES
CN(C(=O)c1ccnn1Cc1ccc2cc(C)c(N)nc2c1)c1ncccc1F
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Compound Formula C21H19FN6O
Compound Structure
Protein Name
Protein arginine N-methyltransferase 5
Protein Classification
Epigenetic regulator
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Writer
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Protein methyltransferase
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Protein arginine methyltransferase
Uniprot ID
O14744
Gene Name
PRMT5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000187 Calu-6 Homo sapiens (Human)  1
1
IC50 = 14 nM
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