Brief Information of the Compound and Protein
Compound Name
 Compound Info 
US8952169, 440
    Show/Hide
 PubChem ID
CID: 86703777
Canonical SMILES
CS(=O)(=O)NC(=O)c1cc(C2CC2)c(OCC2CN(C2)C(c2ccccc2)c2ccccc2)cc1F
    Show/Hide
Compound Formula C28H29FN2O4S
Compound Structure
Protein Name
 Protein Info 
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  2
1
IC50 = 1100 nM
   TI
   LI
   LO
   TS
2
IC50 = 2540 nM
   TI
   LI
   LO
   TS