Brief Information of the Compound and Protein
Compound Name
 Compound Info 
1-[2-[4-(2,4-difluorophenoxy)piperidin-1-yl]-3-[[(3R)-oxolan-3-yl]amino]-7,8-dihydro-5H-pyrido[3,4-b]pyrazin-6-yl]ethanone
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 PubChem ID
CID: 137359492
Canonical SMILES
CC(=O)N1CCc2nc(N3CCC(CC3)Oc3ccc(F)cc3F)c(N[C@@H]3CCOC3)nc2C1
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Compound Formula C24H29F2N5O3
Compound Structure
Protein Name
 Protein Info 
G-protein coupled receptor 6
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
Uniprot ID
P46095
Gene Name
GPR6
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 38000 nM
   TI
   LI
   LO
   TS
CL000308 T-REx-CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 9.4 nM
   TI
   LI
   LO
   TS