Brief Information of the Compound and Protein
Compound Name
6-bromo-2-[(6-chloropyridin-3-yl)methyl]-3,4-dihydropyrazino[1,2-a]benzimidazol-1-one
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PubChem ID
CID: 166633306
Canonical SMILES
Clc1ccc(CN2CCn3c(nc4cccc(Br)c34)C2=O)cn1
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Compound Formula C16H12BrClN4O
Compound Structure
Protein Name
Metabotropic glutamate receptor 2
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q14416
Gene Name
GRM2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000064 Chem-1 Rattus norvegicus (Rat)  1
1
EC50 = 540 nM
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