Brief Information of the Compound and Protein
Compound Name
2-cyclopentyl-4-(5-phenylpyrazolo[1,5-a]pyrimidin-3-yl)benzoic acid
    Show/Hide
Canonical SMILES
OC(=O)c1ccc(cc1C1CCCC1)-c1cnn2ccc(nc12)-c1ccccc1
    Show/Hide
Compound Formula C24H21N3O2
Compound Structure
Protein Name
Calcium/calmodulin-dependent protein kinase kinase 2
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
Other protein kinase group
>
Other protein kinase CAMKK family
>
Other protein kinase Meta subfamily
Uniprot ID
Q96RR4
Gene Name
CAMKK2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 190 nM
   TI
   LI
   LO
   TS
CL000538 LNCaP C4-2 Homo sapiens (Human)  1
1
IC50 = 900 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 21 nM