Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5-[[2,6-difluoro-4-(2-methylindazol-4-yl)phenyl]methyl]-1-(2-methoxyethyl)-4H-pyrrolo[3,4-c]pyrazol-6-one
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 PubChem ID
CID: 146216712
Canonical SMILES
COCCn1ncc2CN(Cc3c(F)cc(cc3F)-c3cccc4nn(C)cc34)C(=O)c12
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Compound Formula C23H21F2N5O2
Compound Structure
Protein Name
 Protein Info 
Muscarinic acetylcholine receptor M1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P11229
Gene Name
CHRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 3930 nM
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