Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-[1-[3-(2-fluoropropan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-4-yl]-6-(1-methylsulfonylpiperidin-4-yl)oxy-N-(trifluoromethyl)pyrimidin-4-amine
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Canonical SMILES
CC(C)(F)c1noc(n1)N1CCC(CC1)N(c1cc(OC2CCN(CC2)S(C)(=O)=O)ncn1)C(F)(F)F
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Compound Formula C21H29F4N7O4S
Compound Structure
Protein Name
 Protein Info 
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q7TQN8
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 24 nM
   TI
   LI
   LO
   TS
CL000657 GLUTag
 Cell Line Info 
Mus musculus (Mouse)  1
1
EC50 = 3.8 nM
   TI
   LI
   LO
   TS