Brief Information of the Compound and Protein
Compound Name
(2S)-6-[(3R)-3-(1-aminocyclopropyl)pyrrolidin-1-yl]-8-cyano-7-fluoro-2-methyl-12-oxo-4-oxa-1-azatricyclo[7.3.1.05,13]trideca-5(13),6,8,10-tetraene-11-carboxylic acid
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PubChem ID
CID: 135369565
Canonical SMILES
C[C@H]1COc2c(N3CC[C@H](C3)C3(N)CC3)c(F)c(C#N)c3cc(C(O)=O)c(=O)n1c23
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Compound Formula C21H21FN4O4
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
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Voltage-gated ion channel
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Potassium channels
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Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 > 30000 nM
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