Brief Information of the Compound and Protein
Compound Name
 Compound Info 
1-[[2-(4-benzylpiperidin-1-yl)-6-(trifluoromethyl)pyridin-3-yl]methyl]-3-(1-oxo-2H-isoquinolin-5-yl)urea
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Canonical SMILES
FC(F)(F)c1ccc(CNC(=O)Nc2cccc3c2cc[nH]c3=O)c(n1)N1CCC(Cc2ccccc2)CC1
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Compound Formula C29H28F3N5O2
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 5.81 nM
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