Brief Information of the Compound and Protein
Compound Name
1-[[2-(3-chlorophenyl)-5-(trifluoromethyl)pyrazol-3-yl]methyl]-3-(1-oxo-2H-isoquinolin-5-yl)urea
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PubChem ID
CID: 66644284
Canonical SMILES
FC(F)(F)c1cc(CNC(=O)Nc2cccc3c2cc[nH]c3=O)n(n1)-c1cccc(Cl)c1
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Compound Formula C21H15ClF3N5O2
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 41.4 nM
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