Brief Information of the Compound and Protein
Compound Name
(R)-2-((cyclopropylmethyl){1-[5'-methyl-2'-(5-oxo-2,5-dihydro-1,2,4-oxadiazol-3-yl)-[1,1'-biphenyl]-4-yl]ethyl}amino)benzo[d]oxazole-4-carboxylic acid
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Canonical SMILES
Cc1ccc(-c2nc(=O)o[nH]2)c(-c2ccc([C@@H](C)N(CC3CC3)c3nc4c(C(=O)O)cccc4o3)cc2)c1
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Compound Formula C29H26N4O5
Compound Structure
Protein Name
Chemerin-like receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Chemokine receptor-like
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Chemerin receptor
Uniprot ID
Q99788
Gene Name
CMKLR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000681 CAL-1 [Human melanoma] Homo sapiens (Human)  2
1
IC50 = 3.2 nM
   TI
   LI
   LO
   TS
2
IC50 = 63 nM
   TI
   LI
   LO
   TS