Brief Information of the Compound and Protein
Compound Name
N-[(1S,2S)-2-hydroxycyclohexyl]-1,6-dimethyl-5-[[4-(1,3-oxazol-4-yl)phenyl]methyl]-2-oxopyridine-3-carboxamide
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Canonical SMILES
Cc1c(Cc2ccc(cc2)-c2cocn2)cc(C(=O)N[C@H]2CCCC[C@@H]2O)c(=O)n1C
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Compound Formula C24H27N3O4
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P11229
Gene Name
CHRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 38 nM
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