Brief Information of the Compound and Protein
Compound Name
1-[(5-tert-butyl-2,3-dihydro-1-benzofuran-2-yl)methyl]-4-prop-2-enylpiperazine
    Show/Hide
Canonical SMILES
CC(C)(C)c1ccc2OC(CN3CCN(CC=C)CC3)Cc2c1
    Show/Hide
Compound Formula C20H30N2O
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
Ki = 15.85 nM
   TI
   LI
   LO
   TS