Brief Information of the Compound and Protein
Compound Name
 Compound Info 
8-[(3R)-3-aminopiperidin-1-yl]-7-but-2-ynyl-3-methyl-1-[3-[4-[5-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl]propyl]purine-2,6-dione
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Canonical SMILES
CC#CCn1c(nc2n(C)c(=O)n(CCCN3CCN(CC3)c3ncc(cn3)C(F)(F)F)c(=O)c12)N1CCC[C@@H](N)C1
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Compound Formula C27H35F3N10O2
Compound Structure
Protein Name
 Protein Info 
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 4020 nM
   TI
   LI
   LO
   TS