Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5,6-dichloro-3-[1-[(4-chlorophenyl)methyl]piperidin-4-yl]-1H-benzimidazol-2-one
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 PubChem ID
CID: 130431397
Canonical SMILES
Clc1ccc(CN2CCC(CC2)n2c3cc(Cl)c(Cl)cc3[nH]c2=O)cc1
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Compound Formula C19H18Cl3N3O
Compound Structure
Protein Name
 Protein Info 
Mu-type opioid receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Opioid receptor
Uniprot ID
P35372
Gene Name
OPRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
EC50 = 15.6 nM
   TI
   LI
   LO
   TS
2
EC50 = 2975 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 1995.26 nM