Brief Information of the Compound and Protein
Compound Name
1-[4-[4-[4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1H-pyrazol-3-yl)amino]pyrimidin-2-yl]phenyl]piperidin-1-yl]prop-2-en-1-one
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PubChem ID
CID: 155804589
Canonical SMILES
CN1CCN(CC1)c1cc(Nc2cc(C)[nH]n2)nc(n1)-c1ccc(cc1)C1CCN(CC1)C(=O)C=C
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Compound Formula C27H34N8O
Compound Structure
Protein Name
Fibroblast growth factor receptor 4
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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TK protein kinase group
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Tyrosine protein kinase FGFR family
Uniprot ID
P22455
Gene Name
FGFR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
GI50 = 438 nM
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