Brief Information of the Compound and Protein
Compound Name
(1S)-1-[2-morpholin-4-yl-4-(trifluoromethyl)phenyl]-N-pyrimidin-2-yl-2,3-dihydro-1H-indene-5-sulfonamide
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PubChem ID
CID: 156010624
Canonical SMILES
FC(F)(F)c1ccc([C@H]2CCc3cc(ccc23)S(=O)(=O)Nc2ncccn2)c(c1)N1CCOCC1
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Compound Formula C24H23F3N4O3S
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 2792 nM
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