Brief Information of the Compound and Protein
Compound Name
(5R,11aS)-2-(2-Fluorophenyl)-5-(4-fluorophenyl)-5,6,11,11a-tetrahydro-1H-imidazo[1',5':1,6]pyrido[3,4-b]-indole-1,3(2H)-dione
    Show/Hide
PubChem ID
CID: 156010507
Canonical SMILES
O=C1[C@@H]2Cc3c([nH]c4ccccc34)[C@@H](c3ccc(F)cc3)N2C(=O)N1c1ccccc1F
    Show/Hide
Compound Formula C25H17F2N3O2
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily M member 8
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
Q8R455
Gene Name
TRPM8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 4400 nM
   TI
   LI
   LO
   TS