Brief Information of the Compound and Protein
Compound Name
(3R,12aS)-3-Benzyl-2,3,12,12a-tetrahydropyrazino-[1',2':1,6]pyrido[3,4-b]indole-1,4(6H,7H)-dione
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PubChem ID
CID: 156021238
Canonical SMILES
O=C1N[C@H](Cc2ccccc2)C(=O)N2Cc3[nH]c4ccccc4c3C[C@@H]12
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Compound Formula C21H19N3O2
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily M member 8
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8R455
Gene Name
TRPM8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 400 nM
   TI
   LI
   LO
   TS