Brief Information of the Compound and Protein
Compound Name
Methyl 3-((1R,3S)-3-((4-Fluorobenzyl)carbamoyl)-2,3,4,9-tetrahydro-1H-pyrido[3,4-b]indol-1-yl)propanoate
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PubChem ID
CID: 156021579
Canonical SMILES
COC(=O)CC[C@H]1N[C@H](C(=O)NCc2ccc(F)cc2)Cc2c1[nH]c1ccccc21
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Compound Formula C23H24FN3O3
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily M member 8
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8R455
Gene Name
TRPM8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 1100 nM
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