Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-cyano-1-[8-[(4-nitro-2,1,3-benzoxadiazol-7-yl)amino]octyl]-3-[3-[3-(1-piperidylmethyl)phenoxy]propyl]guanidine
    Show/Hide
 PubChem ID
CID: 10416230
SID: 15433916
Canonical SMILES
N#CN/C(=N\CCCCCCCCNc1ccc([N+](=O)[O-])c2nonc12)NCCCOc1cccc(CN2CCCCC2)c1
    Show/Hide
Compound Formula C31H43N9O4
Compound Structure
Protein Name
 Protein Info 
Histamine H2 receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Histamine receptor
Uniprot ID
P25102
Gene Name
HRH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000053 COS-7
 Cell Line Info 
Chlorocebus aethiops (Green monkey)  1
1
Ki < 100 nM
   TI
   LI
   LO
   TS