Brief Information of the Compound and Protein
Compound Name
(4S)-1-(2,6-difluoropyridin-4-yl)-5,5-difluoro-3-methylsulfonyl-6,7-dihydro-4H-2-benzothiophen-4-ol
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PubChem ID
CID: 151479053
Canonical SMILES
CS(=O)(=O)c1sc(c2CCC(F)(F)[C@@H](O)c12)-c1cc(F)nc(F)c1
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Compound Formula C14H11F4NO3S2
Compound Structure
Protein Name
Endothelial PAS domain-containing protein 1
Protein Classification
Transcription factor
Uniprot ID
Q99814
Gene Name
EPAS1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000244 786-O Homo sapiens (Human)  1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 < 50 nM