Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-amino-N-[1-(2,5-dichloropyridin-4-yl)azetidin-3-yl]-2,3-dimethylindazole-5-carboxamide
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 PubChem ID
CID: 156011081
Canonical SMILES
Cc1n(C)nc2ccc(C(=O)NC3CN(C3)c3cc(Cl)ncc3Cl)c(N)c12
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Compound Formula C18H18Cl2N6O
Compound Structure
Protein Name
 Protein Info 
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 125 nM
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