Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-amino-2,3-dimethyl-N-[1-[6-(trifluoromethyl)pyridin-3-yl]azetidin-3-yl]indazole-5-carboxamide
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 PubChem ID
CID: 156016090
Canonical SMILES
Cc1n(C)nc2ccc(C(=O)NC3CN(C3)c3ccc(nc3)C(F)(F)F)c(N)c12
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Compound Formula C19H19F3N6O
Compound Structure
Protein Name
 Protein Info 
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 137 nM
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   LI
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