Brief Information of the Compound and Protein
Compound Name
N-[1-(2,5-dichloropyridin-4-yl)azetidin-3-yl]-1-methyltriazolo[4,5-h]quinazolin-6-amine
    Show/Hide
PubChem ID
CID: 156015762
Canonical SMILES
Cn1nnc2ccc3c(NC4CN(C4)c4cc(Cl)ncc4Cl)ncnc3c12
    Show/Hide
Compound Formula C17H14Cl2N8
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 63 nM
   TI
   LI
   LO
   TS