Brief Information of the Compound and Protein
Compound Name
N-[1-(2,5-dichloropyridin-4-yl)azetidin-3-yl]-8,9-dimethylpyrazolo[3,4-h]quinazolin-4-amine
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PubChem ID
CID: 156016190
Canonical SMILES
Cc1n(C)nc2ccc3c(NC4CN(C4)c4cc(Cl)ncc4Cl)ncnc3c12
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Compound Formula C19H17Cl2N7
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 275 nM
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