Brief Information of the Compound and Protein
Compound Name
N-[1-(2,5-dichloropyridin-4-yl)azetidin-3-yl]-3-ethyl-2-methylindazole-5-carboxamide
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PubChem ID
CID: 156016804
Canonical SMILES
CCc1n(C)nc2ccc(cc12)C(=O)NC1CN(C1)c1cc(Cl)ncc1Cl
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Compound Formula C19H19Cl2N5O
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 584 nM
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