Brief Information of the Compound and Protein
Compound Name
N-[1-(5-chloro-2-methoxypyridin-4-yl)azetidin-3-yl]-2,3-dimethylpyrazolo[3,4-c]pyridine-5-carboxamide
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PubChem ID
CID: 156012624
Canonical SMILES
COc1cc(N2CC(C2)NC(=O)c2cc3c(C)n(C)nc3cn2)c(Cl)cn1
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Compound Formula C18H19ClN6O2
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 454 nM
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