Brief Information of the Compound and Protein
Compound Name
2-(3-(4-((4-(1H-Pyrazol-4-yl)phenyl)amino)-6-(tetrahydrofuran-3-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)phenoxy)-N-(tert-butyl)acetamide
    Show/Hide
PubChem ID
CID: 156011037
Canonical SMILES
CC(C)(C)NC(=O)COc1cccc(-c2nc3c(c(Nc4ccc(-c5cn[nH]c5)cc4)n2)CN(C2CCOC2)CC3)c1
    Show/Hide
Compound Formula C32H37N7O3
Compound Structure
Protein Name
Solute carrier family 2, facilitated glucose transporter member 3
Protein Classification
Transporter
>
Electrochemical transporter
>
SLC superfamily of solute carriers
>
SLC02 family of hexose and sugar alcohol transporters
Uniprot ID
P11169
Gene Name
SLC2A3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000134 DLD-1 Homo sapiens (Human)  1
1
IC50 = 155 nM
   TI
   LI
   LO
   TS