Brief Information of the Compound and Protein
Compound Name
2-(3-(4-((4-(1H-Pyrazol-4-yl)phenyl)amino)-6-(1-methoxypropan-2-yl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-2-yl)phenoxy)-N-(tert-butyl)acetamide
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PubChem ID
CID: 156016112
Canonical SMILES
COCC(C)N1CCc2nc(-c3cccc(OCC(=O)NC(C)(C)C)c3)nc(Nc3ccc(-c4cn[nH]c4)cc3)c2C1
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Compound Formula C32H39N7O3
Compound Structure
Protein Name
Solute carrier family 2, facilitated glucose transporter member 1
Protein Classification
Transporter
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Electrochemical transporter
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SLC superfamily of solute carriers
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SLC02 family of hexose and sugar alcohol transporters
Uniprot ID
P11166
Gene Name
SLC2A1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000134 DLD-1 Homo sapiens (Human)  1
1
IC50 = 128 nM
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