Brief Information of the Compound and Protein
Compound Name
2-[3-[6-cyclobutyl-4-[4-(1H-pyrazol-4-yl)anilino]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]phenoxy]-N-(1-methylcyclopropyl)acetamide
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PubChem ID
CID: 156020834
Canonical SMILES
CC1(CC1)NC(=O)COc1cccc(c1)-c1nc2CCN(Cc2c(Nc2ccc(cc2)-c2cn[nH]c2)n1)C1CCC1
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Compound Formula C32H35N7O2
Compound Structure
Protein Name
Solute carrier family 2, facilitated glucose transporter member 1
Protein Classification
Transporter
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Electrochemical transporter
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SLC superfamily of solute carriers
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SLC02 family of hexose and sugar alcohol transporters
Uniprot ID
P11166
Gene Name
SLC2A1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000134 DLD-1 Homo sapiens (Human)  1
1
IC50 = 242 nM
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