Brief Information of the Compound and Protein
Compound Name
N-tert-butyl-2-[3-[6-ethyl-4-[4-(1H-pyrazol-4-yl)anilino]-7,8-dihydro-5H-pyrido[4,3-d]pyrimidin-2-yl]phenoxy]acetamide
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PubChem ID
CID: 124159133
Canonical SMILES
CCN1CCc2nc(nc(Nc3ccc(cc3)-c3cn[nH]c3)c2C1)-c1cccc(OCC(=O)NC(C)(C)C)c1
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Compound Formula C30H35N7O2
Compound Structure
Protein Name
Solute carrier family 2, facilitated glucose transporter member 1
Protein Classification
Transporter
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Electrochemical transporter
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SLC superfamily of solute carriers
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SLC02 family of hexose and sugar alcohol transporters
Uniprot ID
P11166
Gene Name
SLC2A1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000134 DLD-1 Homo sapiens (Human)  1
1
IC50 = 552 nM
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