Brief Information of the Compound and Protein
Compound Name
2-N-(4-chloro-2-methoxy-6-methylphenyl)-4-N-(6-methoxypyridin-3-yl)-3-methyl-4-N-propan-2-ylbenzimidazole-2,4-diamine
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PubChem ID
CID: 155552287
Canonical SMILES
COc1ccc(cn1)N(C(C)C)c1cccc2nc(Nc3c(C)cc(Cl)cc3OC)n(C)c12
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Compound Formula C25H28ClN5O2
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 25 nM
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