Brief Information of the Compound and Protein
Compound Name
N-[2-[4,5-dimethoxy-2-[1-(4-methylphenyl)sulfonylpropyl]phenyl]ethyl]-1-ethyl-6,7-dimethoxy-3,4-dihydro-1H-isoquinoline-2-carboxamide
    Show/Hide
PubChem ID
CID: 122202682
Canonical SMILES
CCC(c1cc(OC)c(OC)cc1CCNC(=O)N1CCc2cc(OC)c(OC)cc2C1CC)S(=O)(=O)c1ccc(C)cc1
    Show/Hide
Compound Formula C34H44N2O7S
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily M member 8
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
Q8R455
Gene Name
TRPM8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
EC50 = 26100 nM
   TI
   LI
   LO
   TS
2
IC50 > 50000 nM
   TI
   LI
   LO
   TS