Brief Information of the Compound and Protein
Compound Name
(3S,11S,14S,22S)-6,8,9,17,19,20-hexamethoxy-7,18-dimethyl-11,22-bis[(E)-2-phenylethenyl]-1,12-diazapentacyclo[12.8.0.03,12.05,10.016,21]docosa-5(10),6,8,16(21),17,19-hexaene-2,13-dione
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PubChem ID
CID: 155567274
Canonical SMILES
COc1c(C)c(OC)c(OC)c2[C@H](\C=C\c3ccccc3)N3[C@@H](Cc12)C(=O)N1[C@@H](Cc2c(OC)c(C)c(OC)c(OC)c2[C@@H]1\C=C\c1ccccc1)C3=O
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Compound Formula C44H46N2O8
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily M member 8
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8R455
Gene Name
TRPM8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 8800 nM
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