Brief Information of the Compound and Protein
Compound Name
4-(2-fluoro-4-furo[3,2-c]pyridin-4-yloxyphenyl)-3,5-dimethyl-1H-pyridazin-6-one
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PubChem ID
CID: 75201899
Canonical SMILES
Cc1n[nH]c(=O)c(C)c1-c1ccc(Oc2nccc3occc23)cc1F
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Compound Formula C19H14FN3O3
Compound Structure
Protein Name
D(1A) dopamine receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Dopamine receptor
Uniprot ID
P21728
Gene Name
DRD1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  3
1
EC50 = 10 nM
   TI
   LI
   LO
   TS
2
EC50 = 490 nM
   TI
   LI
   LO
   TS
3
Ki = 51 nM
   TI
   LI
   LO
   TS